ORIGINAL RESEARCH ARTICLE
ELUCIDATION THE TOXICITY MECHANISM OF METAL OXIDE AND
CARBON-BASED NANOPARTICLES WITH P53 PROTEIN USING
MOLECULAR DOCKING APPROACH
1,
*Krishna Pal Singh,
2
Neeraj Verma and
1,*
Qamar Rahman
1
Amity Institute of Biotechnology, Amity University, Uttar Pradesh, Lucknow, India
2
Society for Biological Research and Rural Development, Kanpur, Uttar Pradesh, India
ARTICLE INFO ABSTRACT
Metal oxide and carbon-based nanoparticles (NP) have a wide range of application in various
fields, including paint, electroluminescent, pharmaceutical, and other industries. In the last
decade, there is an exceeding demand of the applications using these particles in biomedical
sciences such as in drug delivery system whereas these materials are also used widely in the
environmental applications. Due to their extensive applications, these materials are the class of
highest global annual production. The information of the potentially harmful effect of these
nanoparticles lags behind their increased use in consumer products and therefore, the safety data
on various nanoparticles applicable for risk assessment is urgently needed. The availability of less
information of toxicity and harmful effects on the human biological system of these particles,
there is a need to understand the toxicity of metal oxides and carbon-based nanoparticles. In the
present study, we elucidate the toxic impact of the metal oxide and carbon-based nanoparticles on
p53 DNA binding domain protein using molecular docking approach. Furthermore, we also
explore the binding phenomenon between the p53 protein and nanoparticles (metal oxide and
carbon-based NP) using the same molecular docking approach. The study illustrates that metal
oxide based nanomaterial has a high binding affinity toward the DNA binding domain of p53
protein as compared to carbon-based nanoparticles, this happens because the metal oxide
nanoparticles formed hydrogen and metal acceptor bonds whereas in the case of carbon-based
nanoparticles only van der Waal interactions were identified in the molecular interaction. Due to
the binding of these nanoparticles, DNA is unable to interact with binding domain site which may
lead to deactivation of the tumor suppressing nature of the p53 protein.
*Corresponding author:
Copyright©2017, Krishna Pal Singh et al. This is an open access article distributed under the Creative Commons Attribution License, which permits unrestricted
use, distribution, and reproduction in any medium, provided the original work is properly cited.
INTRODUCTION
In recent times, development in nanotechnology engineering
has increased the prompt expansion of many applications for
nanoparticles such as metal nanoparticles (gold, silver etc.),
metal oxide nanoparticles (TiO
2,
CuO, ZnO, fullerene etc.),
C
60
fullerenes nanocrystals, carbon nanotubes (CNTs) in
various industries (Nel et al., 2006; Buzea et al., 2007; De
Stefano et al., 2012; Oberdörster 2012). Principally,
nanoparticles and nanofibers, depict advanced physical and
chemical properties per unit weight, and these activities
explain their vast application not only in industry but also in
the scientific and medical researchers (Jain et al., 2015).
Nanoparticles are unique with their dimensional and structural
properties and extensively been used in various nanomedicine-
related applications, which include cancer targeting,
visualization, and destruction visualization in different
biological systems (Suri et al., 2007; Cai et al., 2008). The
application of nanoparticles as a biomaterial necessitates fully
dissimilar assessments of safety, which include in-silico and
in-vivo analysis, implantation tests, cytotoxicity tests and
carcinogenicity tests, due to the research in last two decades
has highlighted the toxicity and potential risks of their use for
various applications (Hoet et al., 2004; Gangwal et al., 2011;
ISSN: 2230-9926 International Journal of Development Research
Vol. 07, Issue, 08, pp.14449-14454, August, 2017
Article History:
Received 19
th
May, 2017
Received in revised form
17
th
June, 2017
Accepted 10
th
July, 2017
Published online 30
th
August, 2017
Available online at http://www.journalijdr.com
Citation: Krishna Pal Singh, Neeraj Verma and Qamar Rahman, 2017. “Elucidation the toxicity mechanism of metal oxide and carbon-based
Nanoparticles with p53 protein using molecular docking approach”, International Journal of Development Research, 7, (08), 14449-14454.
ORIGINAL RESEARCH ARTICLE Open Access
Keywords:
p53 protein, Metal oxide nanoparticles (TiO2,
ZnO, and CuO), Carbon based nanoparticles
(Fullerene and SWCNT), Molecular docking.