Vol.:(0123456789) 1 3
Chemistry Africa (2021) 4:777–789
https://doi.org/10.1007/s42250-021-00283-3
ORIGINAL ARTICLE
Synthesis and Spectral, Electrochemical, Protein‑Docking
and Biological Studies of Fluoxetine Dithiocarbamate and Its Bivalent
Metal Complexes
Dhananjay Rao Thandra
1
· Venkata Bharat Nishtala
1
· Ramachandraiah Allikayala
1
Received: 15 July 2021 / Accepted: 22 September 2021 / Published online: 29 September 2021
© The Tunisian Chemical Society and Springer Nature Switzerland AG 2021
Abstract
A dithiocarbamate ligand, FLXDTC, has been synthesized from fuoxetine drug along with its complexes of some bivalent
metal ions such as Zn(II), Cd(II), Hg(II), Co(II), Ni(II), Mn(II) and Cu(II). The ligand and the complexes have been charac-
terized by various analytical and spectroscopic methods in addition to some voltammetry studies. The studies propose the
formation M(FLXDTC)
2
complex for all where M = Zn(II), Cd(II), Hg(II), Co(II), Ni(II), Mn(II) and Cu(II) ions. It is also
found that Cu(FLXDTC)
2
takes in more CuCl
2
to result in a Cu
2
(FLXDTC)
2
Cl
2
kind binuclear complex with sulfur atom
bridges Antimicrobial, antioxidant, antifungal, anti-malarial and antitumor capabilities have been tested for both FLXDTC
and M(FLXDTC)
2
complexes. Molecular docking studies on Cu(FLXDTC)
2
with the intercession of EGFR protein show
good antimicrobial and antifungal activities. Biological studies of manganese and nickel complexes have shown excellent anti-
oxidant activity with IC
50
values of 11.29 ± 1.85 and 11.51 ± 1.38 μM. Three diferent cancer cell lines, viz., MCF-7, HepG-2
and HEK 293 have been subjected to the anticancer screening for FLXDTC and it metal complexes whereby it is revealed
that Cd(FLXDTC)
2
has greater activity against MCF-7 (IC
50
= 23.08 ± 0.12 µM), HepG-2 (IC
50
= 12.30 ± 0.25 µM) whereas
Zn(FLXDTC)
2
exhibits good anticancer activity against MCF-7 (IC
50
= 28.63 ± 1.36 µM), HepG-2 (IC
50
= 19.24 ± 1.04 µM).
Extended author information available on the last page of the article