Open Access Research Article
Bari et al., Pharm Anal Acta 2011, 2:2
DOI: 10.4172/2153-2435.1000120
Volume 2 • Issue 2 • 1000120
Pharm Anal Acta
ISSN: 2153-2435 PAA, an open access journal
Keywords: Tamsulosin hydrochloride (TMS); UV-
Spectrophotometry; First order derivative
Introduction
Tamsulosin hydrochloride is a sulphonamide derivative used in the
treatment of Benign Prostate Hyperplasia (BPH), synonymously known
as elders disease.TMS is ofcial in Martindale–Te Extra Pharmacopoeia
and Merck Index [1,2]. TMS, (R)-5-[2-[[2-(2-ethoxyphenoxy)ethyl]
amino]propyl]-2-methoxy-benzenesulfonamide, is a subtype selective
μ
1A
and μ
1D
adrenoceptor antagonist approved by the Food and Drug
Administration (FDA), USA for treatment of BPH. It is a new type of
highly selective α-1-adrenergic receptor antagonist for treatment of
BPH. Compared to other α-antagonists, tamsulosin hydrochloride has
greater specifcity for α-1 receptors in the human prostate and does
not afect receptors on blood vessels. Tamsulosin hydrochloride exists
in two enantiomeric forms but only R-isomer is the pharmaceutically
active component. Literature survey reveals the chiral separation by
electrophoresis [3,4] and HPLC methods, coupled with ESI-MS-MS
are reported for the estimation of tamsulosin hydrochloride with its
impurities in bulk and pharmaceutical formulations [5] as well as in
biological fuids [6-11]. According to our knowledge no method has
been reported for TMS estimation by spectroscopic method. Te
present work deals with estimation of tamsulosin hydrochloride in bulk
and pharmaceutical formulation by simple and derivative spectroscopy
which is economical and intended for better reproducibility of product.
Material and Methods
Chemicals
All reagents used were of analytical grade.
Instrument and conditions
SHIMADZU AUX – 120 (Weighing Balance), UV Shimadzu 2450
(PC Series), UV-visible double beam spectrophotometer, Sofware UV
Probe 2.21, Matched quartz cells 1 cm, Wavelength range 190 -900
nm, Lamp: 50 w, Deuterium Lamp, Detector: Silicon Photodiode, Cell
holder: 1 mm wide, 12 mm high Resolution: 1 nm.
Results and Discussion
Tamsulosin hydrochloride in methanol: water (20:80) solvent
system showed absorbance maximum at 280 nm. In ‘frst order
*Corresponding author: P. S. Jain, R. C. Patel Institute of Pharmaceutical
Education and Research, Karwand Naka, Shirpur-425 405, Dhule (M.S.), Tel: +91
2563 255189; E-mail: pritash79@yahoo.com
Received August 30, 2010; Published April 08, 2011
Citation: Bari SB, Bakshi AR, Jain PS, Surana SJ (2011) Application of UV-
Spectroscopy and First Order Derivative Method for Determination of Tamsulosin
Hydrochloride in Bulk and Tablets. Pharm Anal Acta 2:120.
doi:10.4172/2153-2435.1000120
Copyright: © 2011 Bari SB, et al. This is an open-access article distributed under
the terms of the Creative Commons Attribution License, which permits unrestricted
use, distribution, and reproduction in any medium, provided the original author and
source are credited.
Abstract
Two simple, rapid, sensitive and accurate UV-Spectrophotometry and First order derivative methods have been
developed for estimation of tamsulosin hydrochloride in bulk and tablets. Methanol: water (2:8) was used as a
solvent. In UV spectrophotometric method absorbance of samples are recorded at 280 nm. In frst order derivative
method the amplitude of trough was recorded at 298 nm. Tamsulosin follows linearity in the concentration range of
10-90 μg/ml. Assay results were in good agreement with label claim. These method were validated statistically and
recovery studies.
Application of UV-Spectroscopy and First Order Derivative Method for
Determination of Tamsulosin Hydrochloride in Bulk and Tablets
S. B. Bari, A. R. Bakshi, P. S. Jain*, S. J. Surana
R. C. Patel Institute of Pharmaceutical Education and Research, Karwand Naka, Shirpur-425 405, Dhule (M.S.)
Parameter At 280 nm At 298nm
Linearity equation ( Y= a+ bc ) Y=0.0107X+0.002 0.0046X+ 0.0027
Range(µg/mL) 10.00-90.00 10.00 - 90.00
Correlation Coeffcient(r
2
) 0.9993 0.9977
Table 1: Linear regression data for the calibration curves.
(a)
(b)
Figure 1: Calibration curve for TMS at 280 nm (a) 298 nm (b).
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ISSN: 2153-2435
Pharmaceutica Analytica Acta