Letter to the Editor
The Journal of Clinical Pharmacology
2021, 61(6) 836–837
© 2021, The American College of
Clinical Pharmacology
DOI: 10.1002/jcph.1843
Association Between Baclofen and
Respiratory Depression in Patients With
Chronic Kidney Disease
Satoru Mitsuboshi, PhD
Keywords
adverse event, baclofen, chronic kidney disease, respiratory depression
Baclofen is used to manage spasticity and treat alcohol
use disorder.
1,2
However, because baclofen is eliminated
mainly via the kidneys,
3
users with chronic kidney
disease (CKD) have a high risk of adverse events,
most notably encephalopathy.
4
Respiratory depression
is another serious adverse event caused by baclofen, and
a case report suggested that baclofen caused respiratory
depression in a patient with CKD.
5–7
Although the risk
of respiratory depression caused by baclofen has not
been quantifed, drug-induced respiratory depression
is generally recognized as a serious adverse event that
may even lead to death.
8
In this study, data from
the Japanese Adverse Drug Event Report (JADER)
was used to evaluate whether baclofen increases
the risk of respiratory depression in patients with
CKD.
This was an observational study using anonymized
patient data recorded in JADER, and thus institutional
review board review and approval was not required.
Data recorded from April 2004 to May 2020 were
downloaded from the Pharmaceuticals and Medical
Devices Agency website (http://www.pmda.go.jp/) on
November 3, 2020. Inclusion criteria were all oral
baclofen and eperisone users regardless of whether
the data reporter suspected a possible adverse event.
Eperisone was set as the control because it is used to
manage spasticity. Exclusion criteria were patients who
used both baclofen and eperisone. Patients with missing
data on sex, age, or body weight were also excluded.
Respiratory depression was defned as reporting res-
piratory failure or respiratory depression. CKD was
defned as reporting a comorbidity of CKD, kidney
failure, and use of dialysis. Multiple logistic regression
analysis was used to assess whether use of baclofen
in patients with CKD is a risk factor for respiratory
depression. Sex, age, body weight, and presence of
CKD were considered in the analysis. Modeling was
based on a complete-case analysis. Statistical analysis
was performed using R version 3.4.1 (R Foundation for
Statistical Computing, Vienna, Austria).
In total, 351 baclofen users and 1241 eperisone
users were identifed. Baclofen users with CKD had
a signifcantly increased risk of respiratory depression
(odds ratio, 8.03; 95% confdence interval, 1.88-34.19; P
= .02); no increased risk of respiratory depression was
observed in eperisone users with CKD (Table S1). In
baclofen users, respiratory depression was signifcantly
associated with only the presence of CKD (odds ratio,
7.51; 95% confdence interval, 1.47-38.40; P = .02;
Table 1).
To the author’s knowledge, this is the frst report
to show increased risk of respiratory depression in ba-
clofen users with CKD. Baclofen is eliminated mainly
via the kidneys, and baclofen clearance is equal to cre-
atinine clearance.
9
Therefore, baclofen users with CKD
may have an increased risk of respiratory depression
due to the increased serum concentration of baclofen.
A limitation of this study is potential reporting bias in
JADER, and the results showed increased frequencies
of only certain factors. Respiratory depression is a rare
adverse event; therefore, a clinical trial with a large
sample size would be needed to assess the risk factors.
In conclusion, health care providers should recognize
that baclofen users with CKD are at risk for potential
respiratory depression.
Conficts of Interest
The author declares no conficts of interest.
Funding
No external funding was received to conduct this study.
Department of Pharmacy, Kaetsu Hospital, Niigata, Japan
Submitted for publication 18 January 2021; accepted 19 February 2021.
Corresponding Author:
Satoru Mitsuboshi, PhD, 1459-1 Higashikanazawa, Akiha-ku, Niigata-shi,
Niigata 956-0814, Japan
Email: ccrtyo34057@gmail.com