303
V. V. Holiar, N. Ya. Gotsulyak, A. I. Khoruzhenko
© 2019 V. V. Holiar et al.; Published by the Institute of Molecular Biology and Genetics, NAS of Ukraine on behalf of Bio-
polymers and Cell. This is an Open Access article distributed under the terms of the Creative Commons Attribution License
(http://creativecommons.org/licenses/by/4.0/), which permits unrestricted reuse, distribution, and reproduction in any medium,
provided the original work is properly cited
UDC 576.322, 577.22
Generation and characterization of the MCF-7 cell line with
a knockout of a p85-S6K1 isoform of the ribosomal protein S6 kinase 1
V. V. Holiar, N. Ya. Gotsulyak, A. I. Khoruzhenko, I. V. Zaiets
Institute of Molecular Biology and Genetics, NAS of Ukraine
150, Akademika Zabolotnoho Str., Kyiv, Ukraine, 03143
zaiets.i@gmail.com
Aim. To generate the p85-S6K1 knockout MCF-7 breast cancer cell line and to evaluate the
effect of p85-S6K1 on cell growth, migration and survival under stress conditions. Methods.
CRISPR/Cas9 genome editing, Western blotting, immunofuorescence staining, MTT assay,
in vitro scratch assay. Results. We generated two clones of the p85-S6K1 knockout MCF-7
cell line and tested their survival upon hydrogen peroxide treatment as well as the proliferation
and migration rates. The generated cell clones display an impaired ability to survive under
oxidative stress, exhibit inhibition of cell growth, cell motility and downregulation of rpS6
phosphorylation on Ser235/236/240/244 under cell starvation compared to the control cells.
Conclusions. The p85-S6K1 isoform could be involved in modulation of cancer cell behaviour
promoting cell growth, migration and survival. The obtained clones can be further used to
study the participation of different S6K1 isoforms in the control of cell function.
Keywords: mTOR/S6K1 signaling, CRISPR/Cas9, p85-S6K1 isoform.
Introduction
S6 ribosomal protein kinase 1 (S6K1) is an
extensively studied serine/threonine protein
kinase which functions as a component of the
mTOR/S6K1-dependent signaling pathway. It
is involved in the regulation of protein, lipid
and nucleotide synthesis as well as cell proli-
feration, survival, motility and other cellular
processes (reviewed in [1, 2]). Overactivation
of this kinase leads to the development of a
number of disease states, including obesity,
diabetes and cancer (reviewed in [2–4]). For
example, S6K1 is frequently overexpressed in
breast, lung, ovary, endometrial and thyroid
cancers [5–9]. Its expression correlates with
poor prognosis in patients with breast, kidney
and hepatocellular carcinomas which makes
S6K1 a potential therapeutic target for cancer
treatment (reviewed in [5]). Furthermore, dys-
regulation of mTOR/S6K1 signaling is of spe-
cial signifcance in breast cancer. This signal-
ISSN 1993-6842 (on-line); ISSN 0233-7657 (print)
Biopolymers and Cell. 2019. Vol. 35. N 4. P 303–312
doi: http://dx.doi.org/10.7124/bc.000A0B