American Journal of Molecular Biology, 2022, 12, 135-146
https://www.scirp.org/journal/ajmb
ISSN Online: 2161-6663
ISSN Print: 2161-6620
DOI: 10.4236/ajmb.2022.124012 Aug. 18, 2022 135 American Journal of Molecular Biology
Role of Tyrosine Kinase Receptors in Growth
Factor Mediated Signal Transduction, with
Specific Reference to MAPK/Rasand p13k-Akt
Containing Pathways in Oncogenesis: A
Qualitative Database Review
Chanjugaa Uthayakumar
1
, Rajavarthani Sanjeev
2
1
Trincomalee Campus, Eastern University, Chenkaladi, Sri Lanka
2
Department of Human Biology, Faculty of Health-Care Sciences, Eastern University, Chenkaladi, Sri Lanka
Abstract
Receptor Tyrosine kinases (RTKs) play a crucial role in the signal transduc-
tion pathways at cellular levels. RTK plays a vital role in cellular communica-
tion and transmission of signals to the adjacent cells and regulates different
functions of the cell, such as cellular growth, differentiation, metabolism and
motility. RTK s triggers growth factor receptors such as epidermal growth
factor, insulin growth factor-1 receptor, platelet derived growth factor recep-
tor, and fibro blast growth factor receptor and vascular endothelial growth
factor receptor, thereby initiating and regulating cell growth and prolifera-
tion. MAPK/RAS and PI3/AKT pathways are the major pathways of RTK’s
function. Dysregulation of these RTK’s and pathways often leads to many
diseases such as Noonan Syndrome, Logius Syndrome, CFC syndrome and
different types of cancer. Point mutation and over expression of receptors
and mutations in Ras leads to 30% of human cancers. Also over expression of
different growth factor receptors by RTK too lead to several types of cancers
as Glioblastoma, Thyroid cancer, Colon cancer and Non-small cell lung can-
cer. PTEN mutation in PI3/AKT pathway often leads to carcinoma relative to
Thyroid, Skin, Large intestine, eye and Bone. Therefore, these RTK’s often
used as targets for cancer therapies. The medical sector uses various types of
small molecule tyrosine kinase inhibitors such as ATP competitive inhibitors,
Allosteric inhibitors and covalent inhibitors which are known as Afatinib,
Crizotinib, Eroltinib, Icotinib, Lepatinib and Lenvatinib in treatment and
management of differential carcinomas.
How to cite this paper: Uthayakumar, C.
and Sanjeev, R. (2022) Role of Tyrosine
Kinase Receptors in Growth Factor Me-
diated Signal Transduction, with Specific
Reference to MAPK/Rasand p13k-Akt
Containing Pathways in Oncogenesis: A
Qualitative Database Review. American
Journal of Molecular Biology, 12, 135-146.
https://doi.org/10.4236/ajmb.2022.124012
Received: November 22, 2021
Accepted: August 15, 2022
Published: August 18, 2022
Copyright © 2022 by author(s) and
Scientific Research Publishing Inc.
This work is licensed under the Creative
Commons Attribution International
License (CC BY 4.0).
http://creativecommons.org/licenses/by/4.0/
Open Access