1308 C4H2F2N203 AND CloHvFN203
C(2)--N(1)---C(6) 128.0 (4) C(2)--N(3)---C(4) 125.7 (4)
O(2)----C(2)--N(1) 122.3 (4) O(2)---C(2)--N(3) 122.5 (4)
N(I)----C(2)---N(3) 115.2 (4) O(4)---C(4)--N(3) 122.3 (4)
O(4)----C(4)--C(5) 120.6 (4) N(3)---C(4)--C(5) 117.0 (3)
F(1)---C(5)----C(4) 106.8 (3) F(1)--C(5)--C(6) 106.4 (3)
C(4)---C(5)---C(6) 113.3 (3) F(1)----C(5)---C(7) 108.7 (3)
C(4)----C(5)--C(7) 111.9 (3) C(6)---C(5)----C(7) 109.5 (3)
O(6)---C(6)---N(1) 122.8 (4) O(6)---C(6)---C(5) 121.7 (4)
N(1)---C(6)---C(5) 115.5 (3)
D--H...A D. • .H D. • .A D--H. • .A
o(4i)---H(1).- -N(I~) 2.06 (5) 2.867 (5) 174 (1)
O(6~i)--H(3) .. .N(3 u) 2.00 (5) 2.899 (5) 162 (1)
Symmetry codes: (i) x + ½, ½ - y, -z; (ii) x - ½, ½ - y, -z.
The structures were solved by direct methods and refined
by full-matrix least squares. The non-H atoms were refined
anisotropically; H atoms were located by standard techniques
and were refined isotropically [for (2)], or were placed in
optimized positions (C--H = 0.96~) as a riding model
contribution to the structure-factor calculations [for (1); group
isotropic displacement parameter = 0.08 (2)A2]. Corrections
were applied for Lorentz and polarization effects, and real
and imaginary anomalous dispersion (Cromer, 1974). Structure
solution, refinement and the calculation of derived results were
performed using SHELXTL (Sheldrick, 1986).
Lists of structure factors and anisotropic displacement parameters for
(1) and (2), complete geometry for (2) and packing diagrams for (1)
and (2) have been deposited with the British Library Document Supply
Centre as Supplementary Publication No. SUP 71818 (16 pp.). Copies
may be obtained through The Technical Editor, International Union of
Crystallography, 5 Abbey Square, Chester CH1 2HU, England. [CIF
reference: ST1077]
Acta Cryst. (1994). C50, 1308-1312
Substituted Diphenyl Oxalates
CLIFFORD GEORGE*
Laboratory for the Structure of Matter, Naval Research
Laboratory, Washington DC 20375, USA
P a u l M. LAHTI,* DAVID A. MODARELLI AND
AHMET INCELI
Department of Chemistry, University of Massachusetts,
Amherst, MA 01003, USA
(Received 19 April 1993; accepted 2 November 1993)
Abstract
The ethanedioic acid (oxalic acid) diphenyl ester
derivative with bis(2,6-tert-butyl) substitution, bis-
(2,6-di-tert-butyl-4-methoxyphenyl) ethanedioate,
C32H460 6 (3), adopts an s-trans oxalate conforma-
tion due to steric constraints; such derivatives consti-
tute conformationally well defined molecular
structural units. Diphenyl ethanedioate, C14H1oO4
(1), has approximate s-cis geometry and diphenyl
ethanedioate with tert-butylation on only one ring,
1-(2,4,6-tris-tert-butylphenyl) 2-phenyl ethanedioate,
C26H3404 (2), has a gauche conformation.
References
Bolton, W. (1963). Acta Cryst. 16, 166-173.
Cromer, D. T. (1974). International Tables for X-ray Crystallogra-
phy, Vol. IV, Table 2.3.1. Birmingham: Kynoch Press. (Present
distributor Kluwer Academic Publishers, Dordrecht.)
Cromer, D. T. & Waber, J. T. (1974). International Tables for
X-ray Crystallography, Vol. IV, Table 2.2B. Birmingham:
Kynoch Press. (Present distributor Kluwer Academic
Publishers, Dordrecht.)
DesMarteau, D. D., Resnati, G., Favretto, D. & Traldi, P. (1992).
Org. Mass Spectrom. 27, 204-210.
Harvey, S. C. (1985). Goodman and Gilman's The Pharmacological
Basis of Therapeutics, 7th edition, edited by A. G. Gilman, L. S.
Goodman, T. W. Rail & F. Murad, ch. 17, pp. 339-371. New
York: McMillan.
Larson, A. C. (1970). Crystallographic Computing, edited by F. R.
Ahmed. Munksgaard: Copenhagen.
Meester, P. de, Jovanovic, M. V., Chu, S. S. C. & Biehl, E. R.
(1986). J. Heterocycl. Chem. 23, 337-341.
Resnati, G. (1990a). Farmaco, 45, 1043-1044.
Resnati, G. (1990b). Farmaco, 45, 1137-1139.
Resnati, G. & DesMarteau, D. D. (1992). J. Org. Chem. 57,
4281-4284.
Sheldrick, G. M. (1986). SHELXTL User's Manual. Nicolet XRD
Corporation, Madison, Wisconsin, USA.
Welch, J. T. (1987). Tetrahedron, 43, 3123-3197.
© 1994 International Union of Crystallography
Printed in Great Britain - all rights reserved
Comment
During studies of radical pairs photochemically
generated in neat solid diphenyl ethanedioates (more
commonly called oxalates, a usage we retain in this
work), some of us (Modarelli, George & Lahti, 1991)
wished to study the crystallography of these com-
pounds as a function of different substitution pat-
terns. We found that triplet radical-pair electron-
spirt-resonance (ESR) spectra could be most readily
detected in diphenyl oxalates with 2,6-di-tert-
butylated phenyl rings. More extensive ESR studies
of such radical pairs in oriented crystalline arrays
required definitive structural information. In this
report, we describe the crystal structures and varia-
tion in solid-state molecular conformation of the
following substituted oxalates: diphenyl oxalate (1),
phenyl 2,4,6-tris-tert-butylphenyl oxalate (2) and
bis(2,6-di-tert-butyl-4-methoxyphenyl) oxalate (3).
R) R~
R.~ R~
R2 R"
(i) R,, = R,~ = H
(2) R,, = 'Bu; R,; = H
(3) RI = R2 = R~ = R2 = 'Bu; R3 = R.( = MeO
Acta Co,stallographica Section C
ISSN 0108-2701 ©1994