This is the peer reviewed version of the following article: Feiner, IVJ; Pulagam, KR; Gómez‐ Vallejo, V; Zamacola, K; Baz, Z; Caffarel, MM; Lawrie, CH; Ruiz‐de‐Angulo, A; Carril, M; Ll op, J. Therapeutic Pretargeting with Gold Nanoparticles as Drug Candidates for Boron Neutron Capture Therapy. Part. Part. Syst. Charact.2020, 2000200, which has been published in final form at 10.1002/ppsc.202000200. This article may be used for non-commercial purposes in accordance with Wiley Terms and Conditions for Use of Self-Archived Versions.