Mycoses 2017; 1–5 wileyonlinelibrary.com/journal/myc
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1 © 2017 Blackwell Verlag GmbH
Received: 6 September 2016
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Revised: 11 November 2016
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Accepted: 19 December 2016
DOI: 10.1111/myc.12598
ORIGINAL ARTICLE
Comparatve efcacy of topical applicaton of tacrolimus and
clotrimazole in the treatment of pityriasis versicolor: A single
blind, randomised clinical trial
Mozhdeh Sepaskhah
1
| Maryam Sadat Sadat
1
| Keyvan Pakshir
2
| Zahra Bagheri
3
1
Molecular Dermatology Research Center,
Shiraz University of Medical Sciences,
Shiraz, Iran
2
Basic Sciences in Infectous Diseases
Research Center, Department of Parasitology
and Mycology, School of Medicine, Shiraz
University of Medical Sciences, Shiraz, Iran
3
Department of Biostatstcs, Faculty of
Medicine, Shiraz University of Medical
Sciences, Shiraz, Iran
Correspondence
Mozhdeh Sepaskhah, Molecular Dermatology
Research Center, Shiraz University of Medical
Sciences, Shiraz, Iran.
Email: sepaskhah_m@yahoo.com
Funding informaton
Research deputy of Shiraz University of
Medical Sciences, Grant/Award Number:
91-01-01-5510.
Summary
Background: Pityriasis versicolor (PV) is a common superfcial fungal disease. Possibility
of emergence of resistant strains to azoles, and difculty in diferentaton of hypopig-
mented PV and early vitligo, encouraged us to evaluate the efcacy of topical tacroli-
mus (a calcineurin inhibitor agent with proven in vitro ant-Malassezia efect) for PV
treatment generally and its efect on PV-induced hypopigmentaton specifcally.
Objectves: To evaluate the efcacy of topical tacrolimus on pityriasis versicolor.
Patents/Methods: Fify PV patents were randomly allocated into two equal groups
applying either topical clotrimazol or tacrolimus twice daily for 3 weeks. They were
evaluated at the beginning of study, in the third and ffh weeks clinically and mycologi-
cally (direct smear).
Results: Although both treatments resulted in global, clinical, and mycological cure of
PV, there was no signifcant diference regarding the mentoned aspects of cure be-
tween tacrolimus and clotrimazole treated patents. (P-value: .63, .45, and .26, respec-
tvely) Tacrolimus had no signifcant efect on hypopigmentaton in the ffh week
follow-up. (P-value: .62).
Conclusions: In spite of the lack of efcacy of tacrolimus on PV-induced hypopigmen-
taton, the therapeutc efect on PV introduces tacrolimus as a therapeutc opton for
PV, especially when early vitligo is among the diferental diagnoses without concern-
ing the aggravatng efect of topical cortcosteroids on PV.
KEYWORDS
antfungal agents, clotrimazole, pityriasis versicolor, skin infecton, tacrolimus, treatment, yeast
1 | INTRODUCTION
Malassezia species are involved in the pathogenesis of several skin
disorders.
1
In additon to direct fungal infectons like pityriasis versi-
color and pityrosporum folliculits, Malassezia species are considered
(although controversially in some instances) in the pathogenesis of
some infammatory skin diseases; especially, atopic dermatts, sebor-
rhoeic dermatts and psoriasis.
2
Besides many topical and systemic medicatons tried with vari-
able efcacies to treat Malassezia-associated diseases, including
azole agents (ketoconazole, fuconazole, itraconazole, pramiconazole,
dapaconazole, clotrimazole, miconazole, futrimazole), ciclopirox
olamine, selenium sulphide, adapalene, zinc pyrithione, propylene
glycol and terbinafne,
3–14
in vitro ant-Malassezia efect of calcineurin
inhibitors (tacrolimus and pimecrolimus) has been evaluated.
15,16
Tacrolimus is a macrolide antbiotc discovered as a metabolite of
fungus Streptomyces tsukubaensis. It is a prodrug that afer intracellu-
lar actvaton and combining with FK506-binding protein 12 (FKBP12)
eventually targets calcineurin phosphatase. Calcineurin phospha-
tase dephosphorylates the calcineurin-dependent transcripton fac-
tor (Crz1) and enables it to be translocated into the nucleus where
it actvates the transcripton of genes involved in the regulaton of