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Original article doi: 10.12980/jclm.4.2016J5-230 ©2016 by the Journal of Coastal Life Medicine. All rights reserved.
Degradation study of different brands of paracetamol by UV spectroscopy
Safila Naveed
1*
, Humera Ishaq
2
, Sheeba Urooj
1
1
Faculty of Pharmacy, Jinnah University for Women, Karachi, Pakistan
2
Faculty of Pharmacy, Hamdard University, Karachi, Pakistan
Journal of Coastal Life Medicine 2016; 4(5): 377-379
Journal of Coastal Life Medicine
*Corresponding author: Safila Naveed, Faculty of Pharmacy, Jinnah University for
Women, Karachi, Pakistan.
Tel: +923002621917
E-mail: safila117@yahoo.com, safila117@gmail.com
The journal implements double-blind peer review practiced by specially invited
international editorial board members.
1. Introduction
One of the most common symptoms is pain and this is one
of the most frequent reasons why people seek medical care.
Therefore, it is not surprising that the analgesics are among the
most widely used categories of drug. Hence, for the treatment
of inflammation and pain, paracetamol is used, and chemically
paracetamol (4-hydroxyacetanilide) is used. Paracetamol is a
weak peripheral cycloxygenase inhibitor and from the inhibition
of prostanoid synthesis in the central nervous system, analgesic
effect of paracetamol may arise. Antipyretic effect of paracetamol
is reported to inhibit prostaglandin synthesis at the level of the
hypothalamus causing alteration in body temperature[1].
UV spectrophotometric method used for forced degradation
studies have not been reported in Pakistan. In many laboratories,
spectrophotometric method was used due to less equipment
cost and economical maintenance advantages. By the help of
this technique, the UV absorbance spectra are measured at
200–380 nm. In accordance with the International Conference
on Harmonization guideline, the force degradation state of active
pharmaceutical substance includes acidic, basic and photolytic
conditions. For the estimation of forced degradation of a
pharmaceutical ingredient, acid/base stress testing is performed.
By exposure to acidic or basic medium over time to its chief
degradation products, this test involves degradation of a drug
substance. Acid/base hydrolysis take place in labile carbonyl
functional groups which are amides (lactams), esters (lactones),
aryl amines, imides, imines alcohols and carbamates. The
technique is employed to recognize the raise in the degradation
product and the consequent loss of pharmaceutical active
component i.e. forced degradation is capable to indicate that the
selected technique is a representative of stability[2].
The objective of this study was to analyze forced degradation
studies by treating the different brands of bromazepam under
hydrolytic (acidic and basic), photolytic and thermal stress
ARTICLE INFO ABSTRACT
Objective: To investgate the forced degradation study for the determination of degradation of the
drug substance.
Methods: Paracetamol was exposed to different conditions according to International Conference
on Harmonization guideline. The amount of degradation product can be calculated with the help of
UV spectrophotometer. The official test limits according to British Pharmacopoeia/United States
Pharmacopoeia should not less than and should not more than lapelled amount. Forced degradation
of drug substance was exposed to acidic and basic medium of panadol. Forced degradation of drug
substance of panadol, disprol and calpol were also observed negligible difference in availability on
exposure to UV and heat. This method can be used successfully for studying the stress degradation
factors. Because this method is less time consuming and simple and cost effective also.
Results: The brands i.e. calpol, panadol and disprol, when they come in contact with different
degradation parameters (before, acid, base, heat and UV treatments) according to statistical
analysis, the result showed significant values (P < 0.05) which indicated that there was no
degradation in any of the brand.
Conclusions: The result indicated there is no degradation found in these brands.
Keywords:
Paracetamol
Degradation studies
Different brands
Spectrophotometer
journal homepage: www.jclmm.com
Article history:
Received 19 Nov 2015
Received in revised form 26 Nov, 2nd
revised form 22 Dec 2015, 3rd revised
form 3 May 2016
Accepted 15 May 2016
Available online 20 May 2016