Randomized, Controlled Study of Innovative Spray
Formulation Containing Ozonated Oil and !-Bisabolol
in the Topical Treatment of Chronic Venous Leg Ulcers
Laura Gheuca ˘ Solova ˘stru, MD, PhD; Alina Stı ˆncanu, MD; Alessia De Ascentii, PhD;
Guido Cappare ´, MD; Paolo Mattana; and Dan Va ˆ ¢a ˘, MD, PhD
ABSTRACT
OBJECTIVE: Ozone therapy has a large clinical application in many
therapeutic areas because of its well-known antimicrobial,
immunological, and oxygenating properties. Recently, interest has
grown regarding the application of ozonated oil for vascular leg
ulcer treatment. The efficacy of an innovative spray formulation of
ozonated oil and !-bisabolol combination in the topical treatment
of chronic venous leg ulcers was evaluated compared with standard
epithelialization cream.
DESIGN: A randomized controlled trial was conducted.
SETTING: A total of 29 patients older than 18 years with chronic
venous leg ulcers for less than 2 years’ duration were assessed.
PATIENTS: Patients were randomized to receive daily application
of both ozonated oil and !-bisabolol or the control cream
(vitamin A, vitamin E, talc, and zinc oxide) for 30 days.
MAIN OUTCOME MEASURES: Patients were evaluated on
4 different visits: at days 0, 7, 14, and 30. At each visit, the wound
surfaces were measured. Wound area ratio and the speed of
ulcer healing were calculated.
MAIN RESULTS: At the end of treatment, the proportion of patients
with complete ulcer healing was higher with ozonated oil and !-bisabolol
formulation (25% vs 0%). Furthermore, the changes in ulcer surface
area were significant for ozonated oil and !-bisabolol formulation
only (P G .05), in particular, observing a significant and progressive
reduction of the wound surface by 34%, 59%, and 73%, after 7, 14,
and 30 days of treatment, respectively.
CONCLUSION: The innovative spray formulation of ozonated oil
and !-bisabolol combination shows promise as an important new
therapeutic option in the adjuvant treatment of venous ulcers.
KEYWORDS: !-bisabolol, ozonated oil, topical wound treatment,
venous leg ulcer
ADV SKIN WOUND CARE 2015;28:406Y9
INTRODUCTION
Chronic leg wounds result in diminished quality of life, frequent
hospitalizations and healthcare provider visits, and increased mor-
bidity and mortality.
1
Many leg ulcers are secondary to venous
disease, and epidemiological data presume that approximately 10%
of patients with chronic venous disease develop an ulcer.
2
In addition,
approximately 55% to 70% of all patients with vascular lower-
extremity ulcers have a venous etiology.
3Y5
These data represent
between 0.2% and 1% of the total population and between 1% and
3% of the older adult population in the United States and Europe.
1
Despite various treatment approaches, including the standard
compression therapy, the median duration of an ulcer has been
longer for venous ulcers versus nonvenous ulcers.
6
The healing
time of venous leg ulcers has generally ranged from 40% to 80%
within 3 to 6 months.
3,7,8
Furthermore, venous ulcers are often
recurrent, and open ulcers can persist from weeks to many years.
9
For these reasons, it is important to explore advancements in the
treatment and management of chronic venous ulcers.
Wounds generally follow a well-defined wound healing pro-
cess that involves 4 main stages: coagulation, inflammation, cell
proliferation and repair of the matrix epithelialization, and remod-
eling of the scar tissue.
10
Many studies have demonstrated that endogenous growth fac-
tors, such as fibroblast growth factors,
11
platelet-derived growth
factors,
12
transforming growth factor A,
13
and vascular endothelial
growth factors,
14
are the important regulatory polypeptides in the
healing process. They are released from macrophages, fibroblasts,
and keratinocytes at the site of injury and participate in the reg-
ulation of re-epithelialization, granulation tissue formation, collagen
synthesis, and neovascularization.
From a practical perspective, wound healing depends on many
factors, including wound bed preparation, and the management of
the critical factors summarized in the mnemonic ‘‘TIME’’ framework,
ADVANCES IN SKIN & WOUND CARE & VOL. 28 NO. 9 406 WWW.WOUNDCAREJOURNAL.COM
ORIGINAL INVESTIGATION
Laura Gheuca ˘ Solova ˘ stru, MD, PhD, is Associate Professor, Dermatology Department, Grigore T. Popa University of Medicine and Pharmacy, Iasi, Romania. Alina Stı ˆncanu, MD, is a
Dermatologist, Dermatology, Saint Spiridon Emergency Hospital, Iasi, Romania. Alessia De Ascentii, PhD, is a Scientist, Cosmoproject srl in Casale di Mezzani, and Neovalis srl, Parma,
Italy. Guido Cappare ´ , MD, is a General Practitioner, Lauderma Clinic, Iasi, Romania. Paolo Mattana is a Biologist and Scientific Advisor, Medical Service, Alfa Wassermann, Bologna, Italy.
Dan Va ˆ ¢a ˘, MD, PhD, is Assistant Professor, Dermatology Department, Grigore T. Popa University of Medicine and Pharmacy, Iasi, Romania. Dr Solova ˘stru has disclosed that she was a
consultant for Comsmoproject and was a member of the speakers’ bureau for Pfizer and Berlin Chemie. Paolo Mattana has disclosed that his employer, Alfa Wassermann, is the
pharmaceutical company that markets Azexin (the topical product base of ozonated oil and object of the study). The remaining coauthors have disclosed that they have no financial
relationships related to this article. The authors have disclosed that the article discusses the investigational use of ozonated sunflower oil and !-bisabolol spray formulation in the topical
treatment of chronic venous leg ulcers. Submitted January 21, 2014; accepted in revised form April 15, 2014.
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