_______________________________________________________________________________________________________________________________
3786 https://www.id-press.eu/mjms/index
ID Design Press, Skopje, Republic of Macedonia
Open Access Macedonian Journal of Medical Sciences. 2019 Nov 30; 7(22):3786-3789.
https://doi.org/10.3889/oamjms.2019.504
eISSN: 1857-9655
Herbal Medicine in Pharmaceutical and Clinical Sciences
Cyclin D1, Caspase 9 and P53 Expressions in T47D Cell Lines
after Treatment of Plectranthus amboinicus, (Lour.) Spreng.
Leaves Ethanolic Extract Nanoparticles
Poppy Anjelisa Zaitun Hasibuan
1, 2*
, Sumaiyah Sumaiyah
3
1
Nanomedicine Center of Innovation, Universitas Sumatera Utara, Medan 20155, Indonesia;
2
Departement of Pharmacology
Pharmacy, Faculty of Pharmacy, Universitas Sumatera Utara, Medan 20155, Indonesia;
3
Departement of Technology
Pharmacy, Faculty of Pharmacy, Universitas Sumatera Utara, Medan 20155, Indonesia
Citation: Hasibuan PAZ, Sumaiyah S. Cyclin D1,
Caspase 9 and P53 Expressions in T47D Cell Lines after
Treatment of Plectranthus amboinicus, (Lour.) Spreng.
Leaves Ethanolic Extract Nanoparticles. Open Access
Maced J Med Sci. 2019 Nov 30; 7(22):3786-3789.
https://doi.org/10.3889/oamjms.2019.504
Keywords: Plectranthus ambonicus; Nanoparticle; Cyclin
D1; Caspase-9; p53
*Correspondence: Poppy Anjelisa Zaitun Hasibuan.
Nanomedicine Center of Innovation, Universitas Sumatera
Utara, Medan 20155, Indonesia; Departement of
Pharmacology Pharmacy, Faculty of Pharmacy,
Universitas Sumatera Utara, Medan 20155, Indonesia. E-
mail: poppyanjelisa@usu.ac.id
Received: 25-Sep-2019; Revised: 17-Oct-2019;
Accepted: 18-Oct-2019; Online first: 14-Nov-2019
Copyright: © 2019 Poppy Anjelisa Zaitun Hasibuan,
Sumaiyah Sumaiyah. This is an open-access article
distributed under the terms of the Creative Commons
Attribution-NonCommercial 4.0 International License (CC
BY-NC 4.0)
Funding: This study was supported by Universitas
Sumatera Utara, Indonesia through “Hibah Talenta”
Research Grant 2018 No. 233/UN5.2.3.1/PPM/KP-
TALENTA USU/2018
Competing Interests: The authors have declared that no
competing interests exist
Abstract
BACKGROUND: The application of nanotechnology is aimed to enhance the capability of the chemical
compounds of Plectranthus amboinicus (Lour.) Spreng. leaves activity. The contact area of the particle surface
becomes larger in nano size, which can increase the amount of the isolated active substance. The nanoparticles
of this extract exhibited the most effective impact in decreasing the cell number of T47D by induction of apoptosis
and arresting the cell cycle.
AIM: To evaluate the expressions of cyclin D1, caspase-9 and p53 in T47D cell lines treated by Plectranthus
amboinicus, (Lour.) Spreng. Leaves Ethanolic Extract Nanoparticles (PAEEN).
METHODS: The inhibition of cyclin D1 was done by flow cytometry assay. The expression of cyclin D1, caspase-
9 and p53 were observed by immunocytochemistry assay.
RESULTS: Plectranthus amboinicus, (Lour.) Spreng. Leaves Ethanolic Extract Nanoparticles (PAEEN) on
concentration IC50 (89.2 µg/mL) inhibited the expression of cyclin D1 around 5.59%. Further, the
immunocytochemistry assay indicated that there was an inhibition of cyclin D1, upregulation of caspase-9 and
restoration of p53, indicated by their expression.
CONCLUSIONS: The Plectranthus amboinicus, (Lour.) Spreng. Leaves Ethanolic Extract Nanoparticles could be
an effective anticancer by improving its downregulation on cyclinD1, upregulation caspase-9 and p53.
Introduction
Breast cancer is considered to be one of the
common cancer-related cause of death among
females. Treatment technologies such as surgery,
radiation and chemotherapy are performed by
administering anticancer drugs. Recommended
therapy is the use of compounds from medicinal plant
to reduce the rapid growth of cancer cells [1], [10],
[12].
The cell cycle involves mainly four-step (G1,
S, G2 and M), which lead to cell growth and cell
division to produce two daughter cells. The response
of growth factors in certain cell types is activated by a
complex of CDK-cyclin D [2]. Genetic instability in
cancer cell cause defect in the genes which are
responsible for the checkpoints in the cell cycle.
It has been documented that Plectranthus
amboinicus, (Lour.) Spreng. extract could inhibit the
breast cancer cell by induction of apoptosis and
arresting the cell cycle. The previous study showed
that both single and combination treatment of
Plectranthus amboinicus, (Lour.) Spreng. Ethylacetate
extract 8 μg/mL with doxorubicin 1 μg/mL caused
apoptosis induction and increasing in cell
accumulation at the G1 phase. Expression of cyclin
D1 indicated that both single application and
combination of Plectranthus amboinicus, (Lour.)
Spreng. extract with doxorubicin could arrest the cell
cycle of T47D cells [3].