© 2013 Wichtig Editore - ISSN 0391-3988
Int J Artif Organs ( 2013; : 11) 762-774 36
762
Development and analysis of semi-interpenetrating
polymer networks for brain injection in
neurodegenerative disorders
Marta Tunesi
1,
Sara Batelli
2
, Serena Rodilossi
2
, Teresa Russo
3
, Annalisa Grimaldi
4
, Gianluigi Forloni
2
,
Luigi Ambrosio
3
, Alberto Cigada
1,
Antonio Gloria
3
, Diego Albani
2
, Carmen Giordano
1,
1
Department of Chemistry, Materials and Chemical Engineering “G. Natta”, Politecnico di Milano and Unità di Ricerca
Consorzio INSTM, Politecnico di Milano, Milan - Italy
2
Department of Neuroscience, IRCCS – Istituto di Ricerche Farmacologiche “Mario Negri”, Milan - Italy
3
Institute of Composite and Biomedical Materials, National Research Council of Italy, Naples - Italy
4
Department of Structural and Functional Biology, University of Insubria, Varese - Italy
ORIGINAL ARTICLE
DOI: 10.5301/ijao.5000282
INTRODUCTION
Alzheimer’s (AD) and Parkinson’s diseases (PD) are severe
neurodegenerative disorders strongly linked with aging.
The hippocampus and the entorhinal cortex are the major
brain areas showing the neuropathological lesions of AD,
while in PD the dopaminergic neurons of the substantia
nigra are the most affected, leading to a deficiency of do-
pamine in the striatum. Both diseases significantly impair
the quality of life for patients and their families and their
Purpose: Our aim was to assess the use of injectable, biocompatible and resorbable, hydrogel-based
tools for innovative therapies against brain-related neurodegenerative disorders like Alzheimer’s (AD)
and Parkinson’s (PD) diseases.
Methods: Two compositions of semi-interpenetrating polymer networks (semi-IPNs) based on col-
lagen and poly(ethylene glycol) (PEG) were investigated. We examined their viscoelastic properties,
flow behavior, functional injectability, as well as in vitro biocompatibility with SH-SY5Y human neuro-
blastoma cells and murine primary neurons. We also evaluated the in vivo biological performance after
subcutaneous and brain injection in mice.
Results: The selected semi-IPNs showed a gel-like behavior and were injectable through a 30 G
needle, with the maximum load ranging from 3.0 to 3.9 N. In vitro results showed that immortalized
cells kept their proliferative potential and neurons maintained their viability after embedding in both
materials, with better performances for the gel with the higher collagen content. For both semi-IPNs,
after subcutaneous injection, the inflammatory response was negligible; after brain injection, the tissue
did not show any signs of damage or degeneration.
Conclusions: The results suggest that the selected semi-IPNs not only represent a proper environ-
ment for cells, but also, once injected in vivo, do not induce damage/inflammation in the surrounding
brain tissue. These findings represent a crucial starting point for the development of minimally invasive
and injectable hydrogel-based tools for innovative drug/cell-based therapeutic strategies against AD,
PD, or other severe brain-related neurodegenerative pathologies.
Keywords: Brain, Neurodegenerative diseases, Hydrogels, Semi-interpenetrating polymer networks
Accepted: October 31, 2013