Long-Term Rituximab Use to Maintain Remission of Antineutrophil
Cytoplasmic Antibody–Associated Vasculitis
A Randomized Trial
Pierre Charles, MD; E
´
lodie Perrodeau, MSc; Maxime Samson, MD, PhD; Bernard Bonnotte, MD, PhD; Antoine Ne´ el, MD, PhD;
Christian Agard, MD, PhD; Antoine Huart, MD; Alexandre Karras, MD, PhD; Franc¸ ois Lifermann, MD; Pascal Godmer, MD;
Pascal Cohen, MD; Catherine Hanrotel-Saliou, MD; Nicolas Martin-Silva, MD; Gre´ gory Pugnet, MD, PhD; Franc¸ ois Maurier, MD;
Jean Sibilia, MD, PhD; Pierre-Louis Carron, MD; Pierre Gobert, MD; Nadine Meaux-Ruault, MD; Thomas Le Gallou, MD;
Ste´ phane Vinzio, MD; Jean-Franc¸ ois Viallard, MD, PhD; Eric Hachulla, MD, PhD; Christine Vinter, MD; Xavier Pue´ chal, MD, PhD;
Benjamin Terrier, MD, PhD; Philippe Ravaud, MD, PhD; Luc Mouthon, MD, PhD; and Loı ¨c Guillevin, MD; for the French Vasculitis
Study Group*
Background: Biannual rituximab infusions over 18 months ef-
fectively maintain remission after a “standard” remission induc-
tion regimen for patients with antineutrophil cytoplasmic
antibody–associated vasculitis (AAV).
Objective: To evaluate the efficacy of prolonged rituximab ther-
apy in preventing AAV relapses in patients with granulomatosis
with polyangiitis (GPA) or microscopic polyangiitis (MPA) who
have achieved complete remission after completing an 18-
month maintenance regimen.
Design: Randomized controlled trial. (ClinicalTrials.gov:
NCT02433522)
Setting: 39 clinical centers in France.
Patients: 68 patients with GPA and 29 with MPA who achieved
complete remission after the first phase of maintenance therapy.
Intervention: Rituximab or placebo infusion every 6 months for
18 months (4 infusions).
Measurements: The primary end point was relapse-free sur-
vival at month 28. Relapse was defined as new or reappearing
symptoms or worsening disease, with a Birmingham Vasculitis
Activity Score greater than 0.
Results: From March 2015 to April 2016, 97 patients (mean age,
63.9 years; 35% women) were randomly assigned, 50 to the
rituximab and 47 to the placebo group. Relapse-free survival es-
timates at month 28 were 96% (95% CI, 91% to 100%) and 74%
(CI, 63% to 88%) in the rituximab and placebo groups, respec-
tively, an absolute difference of 22% (CI, 9% to 36%) with a haz-
ard ratio of 7.5 (CI, 1.67 to 33.7) (P = 0.008). Major relapse–free
survival estimates at month 28 were 100% (CI, 93% to 100%)
versus 87% (CI, 78% to 97%) (P = 0.009), respectively. At least 1
serious adverse event developed in 12 patients (24%) in the
rituximab group (with 9 infectious serious adverse events occur-
ring among 6 patients [12%]) versus 14 patients (30%) in the
placebo group (with 6 infectious serious adverse events devel-
oping among 4 patients [9%]). No deaths occurred in either
group.
Limitation: Potential selection bias based on previous rituximab
response and tolerance.
Conclusion: Extended therapy with biannual rituximab infusions
over 18 months was associated with a lower incidence of AAV
relapse compared with standard maintenance therapy.
Primary Funding Source: French Ministry of Health and
Hoffmann–La Roche.
Ann Intern Med. 2020;173:179-187. doi:10.7326/M19-3827 Annals.org
For author, article, and disclosure information, see end of text.
This article was published at Annals.org on 2 June 2020.
* Other investigators and members of the French Vasculitis Study Group
who participated in the study are listed in Supplement 1 (available at
Annals.org).
T
he prognosis of antineutrophil cytoplasmic anti-
body (ANCA)-associated vasculitis (AAV) has dra-
matically improved with the advent of glucocorticoid
treatment and immunosuppressant or rituximab induc-
tion therapy (1). Such regimens lead to remission in 53%
to 88% of patients with AAV (2, 3), but relapse rates re-
main high, making maintenance therapy necessary (4).
Prolonged therapy with azathioprine was once rec-
ommended to maintain AAV remission, because a ran-
domized trial showed lower relapse rates with long-term
azathioprine therapy compared with the standard-length
regimen (5). In 2014, the MAINRITSAN (Maintenance of
Remission Using Rituximab in Systemic ANCA-Associated
Vasculitis) trial reported the clear superiority of rituximab
over azathioprine in maintaining remission (6), which influ-
enced AAV treatment guidelines (7). The therapeutic
schedule of 500 mg of rituximab infused on days 0 and
14, then at months 6, 12, and 18, is now recommended
by the U.S. Food and Drug Administration and European
Medicines Agency to maintain AAV remission. However,
the MAINRITSAN trial showed that relapses after discon-
tinuation of rituximab treatment were frequent, with a
57.9% relapse-free survival rate 32 months after the last
rituximab infusion (8).
The MAINRITSAN3 trial was designed to evaluate
the efficacy of prolonging the rituximab infusion sched-
ule to maintain remission in patients who achieve com-
See also:
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