Vol.:(0123456789) 1 3
Breast Cancer
https://doi.org/10.1007/s12282-018-0894-0
REVIEW ARTICLE
CDKN2A/P16INK4A variants association with breast cancer and their
in-silico analysis
Ayesha Aftab
1
· Shaheen Shahzad
2
· Hafiz Muhammad Jafar Hussain
3
· Ranjha Khan
3
· Samra Irum
1
·
Sobia Tabassum
1
Received: 30 March 2018 / Accepted: 13 July 2018
© The Japanese Breast Cancer Society 2018
Abstract
CDKN2A was first identified as melanoma predisposition tumour suppressor gene and has been successively studied. The
previous researches have not established any noteworthy association with breast cancer. Therefore, through extensive lit-
erature search and in-silico analysis, we have tried to focus on the role of CDKN2A in breast cancer. CDKN2A variants in
breast cancer were collected from different databases. The overall percentage of variants (approximately 5.8%) and their
incidence frequency in breast cancer cases were found to be very low as compared to the number of samples screened in
different studies. Exon 2 was identified as the major region of alternations. Approximately 42.8% were entire gene deletions,
while 24.2% were missense mutations. These variants cannot be ignored because of their pathogenic effects as interpreted by
the bioinformatics tools used in the present study. Earlier studies have shown that CDKN2A excludes the predisposition of
germline variants, but interestingly shares common breast cancer germline variants with other carcinomas. Most of the data
have revealed this gene as rarely mutated or deleted in breast cancer. However, few association studies have shown that in
addition to being a ‘multiple’ tumour suppressor gene, it is mutated/deleted more in breast cancer cell lines as compared to
breast cancer tissues or blood samples; thus, this gene cannot be neglected as a breast cancer candidate gene. The deletion/
malfunctioning of CDKN2A in different tumours including breast cancer has recently led to the discovery of many clinical
CDK inhibitors. Furthermore, these collected genetic variants will also be helpful in developing diagnostic, preventive, and
treatment approaches for patients.
Keywords Breast cancer · Variant analysis · CDKN2A · P16
Introduction
Breast cancer is a type of a tumour in which cancerous
cells originate from tissues of the breast. Males are at fewer
risks of getting breast cancer, but like women, the chances
of developing breast cancer increase with age [1]. It is the
most common cancer in females worldwide with the highest
incidence and mortality rate after lung cancer and has been
ranked second among all of the cancers [1, 2].
In general, two genetic oscillations are involved in tumour
development, one is activation of oncogenes and second
is inactivation of tumour suppressor genes [3]. CDKN2A
(cyclin-dependent kinase inhibitor 2A)/p16INK4A/p14ARF
is an anti-oncogenic or tumour suppressor gene that was
* Shaheen Shahzad
drshaheen@iiu.edu.pk
Ayesha Aftab
ravian09_13@yahoo.com
Hafiz Muhammad Jafar Hussain
hafizaasi19@gmail.com
Ranjha Khan
rhanjha@mail.ustc.edu.cn
Samra Irum
samrairum2@gmail.com
Sobia Tabassum
sobia.tabasum@iiu.edu.pk
1
Department of Bioinformatics and Biotechnology,
International Islamic University, Islamabad 44000, Pakistan
2
Genomics Research Lab, Department of Bioinformatics
and Biotechnology, International Islamic University,
Islamabad 44000, Pakistan
3
The CAS Key Laboratory of Innate Immunity and Chronic
Diseases, School of Life Sciences, University of Science
and Technology of China, Hefei 230027, Anhui, China