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Effect of Florfenicol on Hematology, Cardiac Enzymes and its Residues in Broiler
Chickens by HPLC
Ahmed A. Said
1
, Sameh M. El-Nabtity
1
, Abdulla A.M. Selim
2
, Mai A. Fadel
2*
1
Pharmacology Department, Faculty of Veterinary Medicine, Zagazig University, 44511, Egypt
2
Animal Health Research Institute, Dokki, Giza, Egypt
Article History: Received: 5/3/2016 Received in revised form: 30/5/2016 Accepted: 20/6/2016
Abstract
The current study was conducted on multiple oral doses (40 mg/kg for 3 successive days) of
florfenicol (FF) to determine its effect on some hematological parameters, cardiac enzymes and its
residues in blood and tissues (liver, muscles and kidneys) of broiler chickens. Seventy broiler
chickens were used and divided into two groups, each consisted of 35 birds. The first group was
left as a control, while the second was given FF for 3 successive days. The FF residues in tissues
were determined using reversed phase-high performance liquid chromatography (RP-HPLC)
with ultraviolet (UV) detector at 223 nm. Results indicated a widespread distribution of FF in
most of the tested tissues. All tissue samples were considered FF free on the 9
th
day after the last
oral dose except liver. Florfenicol administration elicited a significant decrease in all blood
parameters (hemoglobin concentration (Hb), red blood cell count (RBCs), mean corpuscular
volume (MCV), mean corpuscular hemoglobin concentration (MCHC) and lymphocytes) from
1
st
up to 7
th
day except packed cell volume (PCV) which showed no significant change on 1
st
day
but decreased on 3
rd
, 5
th
and 7
th
day after stopping medication. Moreover, monocytopenia was
observed on the 5
th
and 7
th
day and white blood cells (WBCs) showed the same effect on the 5
th
day, while heterophiles revealed highly elevation. All cardiac enzymes (aspartate
aminotransferase (AST), lactate dehydrogenase (LDH), creatine kinase MB (CK-MB) and
Troponin I) were highly elevated. In conclusion, broiler chicken meat can be consumed safely
after 9 days post FF treatment.
Keywords: Florfenicol, Broiler chicken, HPLC Residues, Hematological parameters, Cardiac
enzymes
Introduction
Florfenicol (FF) is a bacteriostatic
antibiotic that inhibits protein synthesis by
binding ribosomal subunits of susceptible
bacteria, consequently inhibiting the peptidyl
transferase and then preventing the transfer of
amino acids to growing peptide chains and
subsequent protein formation [1]. Florfenicol
has a fluorine atom instead of the hydroxyl
group located at C-3 in the structure of
chloramphenicol and thiamphenicol. It is used
for treating bovine respiratory disease, in
addition, FF may be considered a bactericidal
against some Mannheimia (Pasteurella)
hemolytica and Pasteurella multocida when it
is administered to achieve minimum
inhibitory concentrations (MICs) [2]. The
minimum bactericidal concentrations (MBCs)
are very close to the MICs.
Following the administration of FF (30
mg/kg BW) in broiler chickens via
intravenous (IV), intramuscular (IM) and oral
routes, the highest drug residues were found
in the kidneys, bile, lungs, muscles, intestine,
heart, liver, spleen and plasma, while the
lowest concentrations were found in brain,
bone marrow and fat [3]. No FF residues were
detected in tissues and plasma after 72 h
except in the bile which disappeared after 96
h [3].
The microbiological Acceptable Daily
Intake (ADI) is 3 μg/kg BW, i.e. 180 μg per
person and a toxicological ADI of 10 μg/kg
BW, i.e. 600 μg per person had previously
been reported by the Committee for
Veterinary Medicinal Products [4]. The
presence of FF residues in broiler meat and
Zagazig Veterinary Journal
Volume 44, Number 1, p. 56-66, June, 2016
©Faculty of Veterinary Medicine, Zagazig University, 44511, Egypt
DOI: 10.21608/zvjz.2016.7832.
*Corresponding author e-mail: (dr.mai87@yahoo.com), Animal Health Research Institute, Dokki,
Giza, Egypt.