International Journal of Pharmaceutical Chemistry and Analysis 2024;11(1):85–90
Content available at: https://www.ipinnovative.com/open-access-journals
International Journal of Pharmaceutical Chemistry and
Analysis
Journal homepage: https://www.ijpca.org/
Original Research Article
Design, formulation and in-vitro evaluation of diclofenac sodium fast
disintegrating tablets
P SS Prasanna Kumar
1
*, T Anjali
1
, Srinivas Nandyala
2
, K. Sivaji
1
1
Dept. of Pharmaceutics, A.K.R.G College of Pharmacy, Nallajerla, Andhra Pradesh, India
2
Dept. of Pharmacology, A.K.R.G College of Pharmacy, Nallajerla, Andhra Pradesh, India
ARTICLE INFO
Article history:
Received 10-02-2024
Accepted 13-03-2024
Available online 26-03-2024
Keywords:
Diclofenac sodium
NSAID
Zea mays L (Corn silk) extract powder
Fast disintegrant
ABSTRACT
Diclofenac sodium is an agent shows Anti-Inflammatory, Anti-pyretic and Analgesic activity. The present
work of the study is to design, formulate a tablet by using powder from Corn silk which disintegrate,
dissolve rapidly, thereby gives rapid onset of action and investigate the fast-disintegrating property. The
natural polymer chosen for the purpose of study is due to disintegrating property, non-toxicity, low
cost, reliable, free availability, eco-friendly, potentially degradable and compatible. The formulation has
been prepared" Corn silk " powder with various 05 different concentrations 2-10%W/W using direct
compression method and evaluations are conducted. Each formulation has been Evaluated for various
parameters of pre and post compression tablets namely Bulk density, tapped density, Angle of repose,
Weight variation, Hardness, Friability, Wetting time, Disintegration time, In- vitro dissolution studies. The
in vitro dissolution studies revealed that F5 with 10%w/w of Corn silk achieved a remarkable release of
99.98% of the drug within 25 minutes.
The inclusion of corn silk in F5 significantly enhances the dissolution rate of diclofenac sodium compared
with other formulations.
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1. Introduction
Drug delivery is the most important and vastly
using technique for administration of an API to
show pharmacological activity, achieve a therapeutic
effect, primarily due to patient acceptability, ease of
administration, inexpensive manufacturing process and
release pattern. For many drugs, tablets incorporated with
rapid disintegrating agent provide clinically effective
treatment thereby maintains the required balance of
pharmacokinetic and pharmacodynamic profiles of API
with acceptable levels of patient safety and efficacy. These
API and excipients are designed to formulate and to provide
* Corresponding author.
E-mail address: pssprasanna1@gmail.com (P. S. S.
Prasanna Kumar).
maximum stability, activity and bioavailability.
1
Fast disintegrating tablets are those that disintegrate
rapidly and release the drug by dissolving. A disintegrant
is belongs to the tablet excipient, and it was incoeporated
to dosage form which we have chosen either it maybe
a tablet or capsule for breakup of the compacted
mass when it is enter into a fluid environment(gastric
fluid or intestine).
2
Disintegrants are added to tablets
or encapsulated formulations to break the tablet or
capsule slugs into smaller fragments in the presence
of solvent(aqueous) environment, thereby increasing the
available particle surface area promote API to release more
rapidly.
3,4
https://doi.org/10.18231/j.ijpca.2024.012
2394-2789/© 2024 Author(s), Published by Innovative Publication. 85