Intensive Care Med (2004) 30:1690–1691
DOI 10.1007/s00134-004-2335-0
(HR 90/min, day 12) while the QRS com-
plex always remained less than 12 ms.
The patient was becoming progressively
more agitated and as this was interpreted
as probable methadone withdrawal, meth-
adone was reintroduced on day 12 at a
dose of 130 mg per day. On the next day
the QTc interval started gradually increas-
ing. It rose to 552 ms (HR 83/min) on the
next day (day 13) and reached 581 ms
(HR 91/min) on day 19. Given the poor
prognosis, further resuscitation efforts
were deemed futile, and the patient died
2 days later from ventilator associated
pneumonia.
Methadone is a synthetic opioid widely
used for the treatment of narcotic addic-
tion. Tolerance may develop, and the daily
maintenance dose must be increased in
patients treated by oral methadone for sev-
eral years. Until recently there was little
evidence of the effect of methadone on the
human heart. Kornick et al. [5] found in
patients treated by intravenous methadone
for cancer pain that there is an approxi-
mately linear relationship between QTc
interval prolongation and the log-dose of
methadone. In these patients the presence
of chlorbutanol in the commercial solution
was considered a possible contributing fac-
tor. However, the authors were demonstra-
ted that methadone alone blocked cardiac
human ether a-go-go related gene (HERG)
K
+
channels in vitro in comparable concen-
trations to those observed in the patients
receiving intravenous methadone for
chronic pain management. A prospective
study conducted in 132 drug-addicted
patients beginning oral methadone main-
tenance treatment observed a significant
increase in the QTc interval between base-
line and follow-up [4]. Men and patients
receiving higher methadone doses
(110–150 mg) had the greatest prolonga-
tion. Gil et al. [1] recently found that
four patients infected with the human
immunodeficiency virus developed syn-
cope and prolongation of the QT interval
while receiving high doses of methadone
(>200 mg/day); shortening of the QT inter-
val occurred when methadone doses were
reduced.
Among the other drugs or substances
taken by our patient, fluoxetine, olanzap-
ine, and cocaine can also cause QT interval
prolongation and may be associated with
torsades de pointes. The hallmark of co-
caine intoxication is wide complex arrhyth-
mia which was absent in our patient [6].
Fluoxetine can cause QTc prolongation in
toxic doses. Three clinical studies involv-
ing 350 patients treated with fluoxetine
showed no significant changes in the QTc
interval. There is a single case report of
QTc prolongation in a patient taking 40 mg
fluoxetine daily which resolved after fluox-
etine was stopped. Our patient was taking
half of that dose and had therapeutic flu-
oxetine levels on admission. Additionally
the QTc prolongation reappeared despite
the discontinuation of fluoxetine [7, 8].
Therapeutic olanzapine and trazodone have
mild and clinically nonsignificant effects
on QTc prolongation [9, 10].
The QTc interval showed a dose-re-
sponse relationship consistent with the
administration of methadone; it gradually
decreased when methadone was stopped
and became immediately prolonged after
methadone was reinstituted. Our patient
had a normal QTc interval 4 years prior to
the event while he was taking the same
amount of methadone (404 ms vs. 576 ms
postresuscitation). The delayed effect of
methadone on the QTc interval and ques-
tionable compliance of the patient can
probably explain this difference. Although
cocaine may have contributed to our
patient’s cardiac arrest, we believe that
this effect took place on an already com-
promised heart secondary to the document-
ed QTc prolongation induced by metha-
done. This effect was reported to the local
drug safety center.
In conclusion, in addition to the experi-
mental evidence supporting the concept
that methadone prolongs the QTc interval
through a dose-dependent mechanism,
there is an increasing number of reports
suggesting that this effect can also occur
in humans. Consequently the QT interval
should be carefully monitored especially
when the dose of methadone is increased
or when the patient is given other medica-
tions which could also affect the QT inter-
val [11].
References
1. Gil M, Sala M, Anguera I, Chapinal O,
Cervantes M, Guma JR, Segura F
(2003) QT prolongation and torsades
de pointes in patients infected with
human immunodeficiency virus and
treated with methadone. Am J Cardiol
92:995–997
2. Lipski J, Stimmel B, Donoso E (1973)
The effect of heroin and multiple
drug abuse on the electrocardiogram.
Am J Heart 86:663–668
3. Krantz MJ, Lewkowiez L, Hays H,
Woodroffe MA, Robertson AD, Mehler
PS (2002) Torsade de pointes associat-
ed with very-high-dose methadone.
Ann Intern Med 137:501–504
4. Martell BA, Arnsten JH, Ray B,
Gourevitch MN (2003) The impact
of methadone induction on cardiac
conduction in opiate users. Ann Intern
Med 139:154–155
CORRESPONDENCE
J. A. Decerf
B. Gressens
C. Brohet
A. Liolios
P. Hantson
Can methadone prolong
the QT interval?
Accepted: 10 May 2004
Published online: 8 June 2004
© Springer-Verlag 2004
Sir: The cardiac safety of high doses of
methadone has been questioned in recent
publications describing the impact of meth-
adone on cardiac conduction [1, 2, 3, 4].
We present a case of prolonged QTc inter-
val in a patient treated with methadone for
several years.
A 37-year-old man was found in cardiac
arrest (asystole) and was successfully
resuscitated. He had been receiving
methadone maintenance treatment for
more than 8 years at a daily oral dose of
130 mg; it is not known how compliant
the patient was during these years. Elec-
trocardiography (ECG) performed in 2000
while the patient was on methadone re-
vealed sinus bradycardia (49/min) with a
normal QRS interval and a normal QTc
interval of 404 ms. The patient was also
taking fluoxetine (20 mg/day), trazodone
(10 mg/day), and olanzapine (5 mg/day).
According to his wife, he had used co-
caine (“sniffing”) a few hours before the
cardiac arrest, but he was not seen taking
an excessive dose of methadone. Toxico-
logical screening showed therapeutic
serum levels of fluoxetine, trazodone,
and olanzapine, and the presence in the
patient’s serum of two cocaine metabo-
lites [benzoylecgonine (0.263 μg/ml),
methylecgonine (0.012 μg/ml)] and meth-
adone (0.229 μg/ml). Postresuscitation
ECG showed sinus rhythm (90/min) with
a QRS complex less than 100 ms and a
QTc interval of 576 ms; there were no
findings consistent with ischemia. No
electrolyte abnormalities were noted. The
patient developed anoxic encephalopathy
with a poor prognosis for neurological re-
covery. The only medication the patient
was receiving was low doses of propofol
for fighting the ventilator. ECG changes
were monitored daily. Methadone and
its metabolites were still detected in the
blood until day 7 and in the urine until
day 11. Cocaine metabolites were detected
in the serum until day 4. The QTc inter-
val gradually decreased from 600 ms
(heart rate, HR, 72/min, day 2) to 485 ms