© Asian Journal of Biomedical and Pharmaceutical Sciences, 2016.
e Effect of the Antioxidant Drug “U-74389G” On Oviductal Congestion during
Ischemia Reperfusion Injury in Rats
e effect of the antioxidant drug “U-74389G” was examined, on rat model and particu-
larly in an oviductal ischemia reperfusion (IR) protocol. e probable effects of that mole-
cule were studied pathologically using oviductal congestion (OC) lesions. 40 rats of mean
weight 231.875 g were used in the study. OC lesions were evaluated at 60 min of reperfusion
(groups A and C) and at 120 min of reperfusion (groups B and D) in rats. U-74389G was
administered only in groups C and D. U-74389G administration non-significantly altered
the OC scores by 0 without lesions [-0.3582422 - 0.3582422] (p=0.9608). Reperfusion time
non-significantly increased the OC scores by 0.2 without lesions [-0.1521699 - 0.5521699]
(p= 0.2317). However, U-74389G administration and reperfusion time together signifi-
cantly increased the OC scores by 0.0909091 without lesions [-0.1230462 - 0.3048644]
(p=0.3951). U-74389G administration whether it interacted or not with reperfusion time
failed to restore the OC lesions within short-term time context of 2 hours.
Keywords: ischemia; U-74389G; fallopian tubes; oviductal congestion; reperfusion
ABSTRACT :
Tissue ischemia and reperfusion (IR) are among the
main causes of permanent or transient damage with
serious implications on adjacent organs and certainly on
patients’ health. e usage of antioxidant substances as
a treatment is a new concept. Furthermore, satisfactory
answers have not been given yet to fundamental
questions, such as, how fast does U-74389G act, when
should U-74389G be administered, and at what dosage.
e particularly satisfactory action of the antioxidant
U-74389G in tissue protection has been noted in several
performed experiments. Aſter a careful literature search
was conducted, it was realized that this certain antioxidant
has been tried in IR experiments. However, just few
relative reports were found, not covering completely this
particular matter. Also, many publications addressed trials
of other similar molecules of aminosteroids (lazaroids) to
which the studied molecule also belongs to. U-74389G
or better 21-[4-(2,6-di-1-pyrrolidinyl-4-pyrimidinyl)-1-
piperazinyl]-pregna-1,4,9(11)-triene-3,20-dione maleate
salt is an antioxidant which prevents both arachidonic
acid-induced and iron-dependent lipid peroxidation
[www.caymanchem.com]. It protects against IR injury in
animal heart, liver and kidney models. ese membrane-
associating antioxidants are particularly effective in
preventing permeability changes in brain microvascular
endothelial cells monolayers [Fenglin et al., 1995]. A meta-
analysis of 13 published seric variables, coming from the
same experimental setting, tried to provide a numeric
evaluation of U-74389G efficacy at the same endpoints
(Table 1).
e aim of this experimental study was to examine the
effect of U-74389G on rat model and particularly in an
oviductal IR protocol. e probable effects of that molecule
were studied by evaluating the oviductal congestion (OC)
lesions.
MATERIALS AND METHODS
Animal preparation
is experimental study was licensed by the Veterinary
Address of East Attiki Prefecture under 3693/12-11-2010
& 14/10-1-2012 decisions. It was done at the Experimental
Research Centre of ELPEN Pharmaceuticals Co. Inc.
S.A. at Pikermi, Attiki. Everything needed for the study
*Corresponding author:
Constantinos Tsompos
Department of Obstetrics & Gynecology, Mesologi County Hospital, Etoloakarnania, Greece
Email: Constantinostsompos@yahoo.com
doi: 10.15272/ajbps.v6i52.765
INTRODUCTION:
Received on:06/12/2015
Accepted on: 10/01/2016
Published on: 23/01/2016
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Article Info:
O pen A ccess
Literati
Research Article
Constantinos Tsompos
1*
, Constantinos Panoulis
2
, Konstantinos Toutouzas
3
, George Zografos
3
, Apostolos Papalois
4
1
Department of Obstetrics & Gynecology, Mesologi County Hospital, Etoloakarnania, Greece
2
Department of Obstetrics & Gynecology, Aretaieion Hospital, Athens University, Attiki, Greece
3
Department of Surgery, Ippokrateion General Hospital, Athens University, Attiki, Greece
4
Exprerimental Research Center ELPEN Pharmaceuticals, S.A. Inc., Co., Attiki Greece
Conflict of interest: Authors reported none
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