J vet Pharmacol Therap. 2018;1–5. wileyonlinelibrary.com/journal/jvp
|
1 © 2018 John Wiley & Sons Ltd
Thiamphenicol (TP) and its fluorinated derivative florfenicol (FF)
are antimicrobials widely used in veterinary medicine. They act by
binding to the 50S ribosomal subunit, leading to inhibition of pro-
tein synthesis and bacteriostatic effect. FF and TP are used in a
broad spectrum of infections caused by, for example., Pasteurella
multocida, Staphylococcus aureus, Haemophilus sp., Bacteroides sp.,
and Streptococcus sp. in companion animals, farm animals and fish
(Beers, Schoutens, Vanderlinden, & Yourassowsky, 1975; Switala &
Debowy, 2005; Wei, Shien, Chang, & Chou, 2016; Wei et al., 2016;
Yoshimura, Takagi, Ishimura, & Endoh, 2002).
Pharmacokinetics (PK) of these two agents were described in
cattle (Abdennebi, Sawchuk, & Stowe, 1994; Varma, Adams, Powers,
Powers, & Lamendola, 1986), pigs (Haritova, Lashev, & Pashov,
2002; Jiang, Zeng, Chen, Liu, & Fung, 2006), rabbits (Abd El-Aty,
El-Sooud, & Goudah, 2001; Park, Lim, Kim, Hwang, & Yun, 2007),
dogs (Castells et al., 1998; Park, Lim, Kim, Hwang, & Yun, 2008),
and sheep (Abdennebi, Khales, Sawchuk, & Stowe, 1994; Jianzhong,
Xiubo, Haiyang, & Walter, 2004). As for birds, the scientific literature
is rich in studies on FF PK in chickens (Afifi & Elsooud, 1997; Chang
et al., 2010; Shen, Hu, Wu, & Coats, 2003) and turkeys (Switala et al.,
2007; Watteyn, Croubels, De Baere, De Backer, & Devreese, 2018).
Ismail and El-Kattan (2009) investigated FF kinetics in pigeons and
quail while El-Banna (1998) assessed it in healthy and Pasteurella-
infected ducks following intravenous (IV) and intramuscular injec-
tion. The latter study, however, was carried out using microbiological
assay which has significant drawbacks compared with chromato-
graphic techniques (Marzo & Dal Bo, 1998). The literature on TP in
poultry is limited to PK in chickens (Chen & Pu, 2008) and turkeys
(Switala et al., 2007). There are no available data on TP PK in ducks.
Considering physiological differences between waterfowl and other
birds (Dorrestein & Vanmiert, 1988), it seems that simple extrapola-
tion of dosage protocols from terrestrial birds to ducks may not be
justified. Therefore, the aim of the study was to compare FF and TP
PK in ducks after single IV and oral (PO) administration.
Received: 23 May 2018
|
Revised: 8 August 2018
|
Accepted: 22 August 2018
DOI: 10.1111/jvp.12714
SHORT COMMUNICATION
Pharmacokinetics of florfenicol and thiamphenicol in ducks
Marta Tikhomirov | Błażej Poźniak | Andrzej Smutkiewicz | Marcin Świtała
Department of Pharmacology and
Toxicology, Faculty of Veterinary
Medicine, Wrocław University of
Environmental and Life Sciences, Wrocław,
Poland
Correspondence
Marta Tikhomirov, Department of
Pharmacology and Toxicology, Faculty of
Veterinary Medicine, Wrocław University of
Environmental and Life Sciences, Wrocław,
Poland.
Email: marta.tikhomirov@upwr.edu.pl
Funding information
Ministry of Science and Higher Education of
the Republic of Poland – KBN, Grant/Award
Number: 3 PZ6K 03724
Abstract
The pharmacokinetics of florfenicol (FF) and thiamphenicol (TP) after single intrave-
nous (IV) and oral (PO) administration was investigated in Mulard ducks. Both antibi-
otics were administered at a dose of 30 mg/kg body weight, and their concentrations
in plasma samples were assayed using high-performance liquid chromatography with
ultraviolet detection. Pharmacokinetic parameters were calculated using a noncom-
partmental method. After IV administration, significant differences were found for
the mean residence time (2.25 ± 0.21 hr vs. 2.83 ± 0.50 hr for FF and TP, respec-
tively) and the general half-life (1.56 ± 0.15 hr vs. 1.96 ± 0.35 hr for FF and TP, re-
spectively) indicating slightly slower elimination of TP as compared to FF. The
clearance, however, was comparable (0.30 ± 0.07 L/hr/kg for FF and 0.26 ± 0.04 L/
hr/kg for TP). The mean volume of distribution was below 0.7 L/kg for both drugs.
Pharmacokinetics after PO administration was very similar for FF and TP suggesting
minor clinical importance of the differences found in the IV study. Both antimicrobi-
als showed rapid absorption and bioavailability of more than 70% indicating that PO
route should be an efficient method of FF and TP administration to ducks under field
conditions.
KEYWORDS
antimicrobials, ducks, florfenicol, pharmacokinetics, thiamphenicol