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International Journal of Chemical Studies 2025; 13(4): 102-106
P-ISSN: 2349–8528
E-ISSN: 2321–4902
www.chemijournal.com
IJCS 2025; 13(4): 102-106
© 2025 IJCS
Received: 09-04-2025
Accepted: 13-05-2025
SP Soul Shekhar
Department of Chemistry, Guru
Nanak First Grade College,
Bidar, Karnataka, India
ND Satyanarayan
Department of Pharmaceutical
Chemistry, Kuvempu
University, Post Graduate
Centre, Kadur, Karnataka, India
CH Chandrashekhar
Department of Pharmaceutical
Chemistry, Kuvempu
University, Post Graduate
Centre, Kadur, Karnataka, India
Corresponding Author:
SP Soul Shekhar
Department of Chemistry, Guru
Nanak First Grade College,
Bidar, Karnataka, India
Α-amylase inhibitory potential of Balanites
roxburghiana Linn. fruit extracts: A comparative
solvent-based study
SP Soul Shekhar, ND Satyanarayan and CH Chandrashekhar
DOI: https://www.doi.org/10.22271/chemi.2025.v13.i4b.12564
Abstract
The global prevalence of diabetes mellitus necessitates the exploration of novel therapeutic interventions
with minimal adverse effects. This research evaluates the enzyme inhibitory properties of Balanites
roxburghiana fruit extracts against α-amylase using three different solvents (n-hexane, dichloromethane,
and methanol) through chromogenic DNSA methodology. The investigation revealed remarkable
variance in bioactivity among solvent extracts. n-hexane extract exhibited exceptional inhibitory
capacity, demonstrating concentration-responsive effects with maximum inhibition of 90.10% at 500
μg/mL, followed by 62.03% and 51.52% at 250 and 100 μg/mL respectively. Dichloromethane extract
showed limited bioactivity (4.86-7.29%), while methanol extract unexpectedly enhanced enzymatic
activity. Acarbose served as reference standard with complete inhibition across all concentrations.
Phytochemical evaluation identified steroids and saponins as predominant compounds in the active n-
hexane fraction. These outcomes establish the therapeutic significance of lipophilic constituents in B.
roxburghiana fruits for managing postprandial hyperglycemia.
Keywords: Antidiabetic agents, Balanites roxburghiana, Enzyme inhibition, Natural products,
Postprandial glucose control, Chromogenic assay
1. Introduction
The escalating global burden of metabolic disorders, particularly type 2 diabetes mellitus,
presents unprecedented challenges to healthcare systems worldwide. This chronic condition
affects approximately 537 million adults globally, with projections indicating continued
growth due to lifestyle modifications and demographic transitions. The pathophysiological
complexity involves multiple defects including impaired insulin secretion, peripheral insulin
resistance, and dysregulated hepatic glucose metabolism
[1]
. Contemporary therapeutic
approaches rely heavily on synthetic pharmaceuticals, including metformin, sulfonylureas, and
α-glucosidase inhibitors. However, these interventions frequently produce undesirable
complications such as gastrointestinal dysfunction, weight gain, and hypoglycemic episodes
[2]
.
The limitations of existing treatments have catalyzed research into plant-derived alternatives
that may offer superior safety profiles with comparable efficacy. Enzymatic carbohydrate
digestion represents a critical regulatory point for glucose homeostasis. α-Amylase, a key
digestive enzyme, catalyzes the initial breakdown of complex carbohydrates into
oligosaccharides and simple sugars. Therapeutic intervention at this level can effectively
modulate postprandial glucose excursions without inducing severe hypoglycemia
[3]
. This
approach has gained considerable attention as a promising strategy for diabetes management.
1.1 Botanical Profile and Ethnobotanical Significance
Balanites roxburghiana Planch. (Zygophyllaceae) represents a taxonomically significant
species indigenous to arid ecosystems across Africa and South Asia. This xerophytic plant
exhibits remarkable environmental adaptability, thriving in harsh climatic conditions where
conventional vegetation fails to survive. The species displays characteristic morphological
features including thorny branches, compound leaves, and distinctive elongated fruits
[4, 5]
.
Traditional medicine systems have extensively utilized various plant parts for treating diverse
ailments. Historical records document its application in managing metabolic disorders,
inflammatory conditions, and infectious diseases. Contemporary ethno botanical surveys
continue to validate traditional knowledge, revealing ongoing utilization by indigenous
communities across its natural distribution range.