*Corresponding Author Address: Hardik Makwana, Parul Institute of pharmacy, Vadodara, India; Email id:
hardik_makwana58@ymail.com
World Journal of Pharmaceutical Sciences
ISSN (Print): 2321-3310; ISSN (Online): 2321-3086
Published by Atom and Cell Publishers © All Rights Reserved
Available online at: http://www.wjpsonline.org/
Original Article
Formulation, optmization and evaluation of taste masked oral disintegrating tablet of
verapamil HCL
Hardik Makwana
1*
, Parag Patel
1
, Prashant Patel
2
, Bhawankumar P. Patel
3
1
Parul Institute of pharmacy, Limda, Vadodara, India
2
Mercury laboratories limited, Vadodara, India
3
Rowan University, Glassboro, NJ.08028
Received: 29-04-2015 / Revised: 18-05-2015 / Accepted: 20-05-2015
ABSTRACT
Verapamil HCl is calcium channel blocker used for the treatment of hypertension, irregular heartbeat, angina,
and to control the systolic and diastolic blood pressure. As Verapamil HCl is bitter in taste, taste masking is
required for preparing oral disintegrating tablet. To mask the taste we used resin Indion 234. Oral disintegrating
Tablets were made using various superdisintegrants (crosspovidone, SSG, Kyron T 314) at 3 different
concentration with three different ratio (Drug: Indion 234) 1:1, 1:2, 1:3 of drug and resin equivalent to 40mg
form a Drug Resin complex (DRC). Crosspovidone shows the best disintegration time and it is further used for
the formulation of the tablets. All the formulations were evaluated for parameters such as hardness, friability,
disintegration time, in vitro drug release. An effective formulation F8 having hardness 4.1 kg/cm
2
,
disintegration time of 21sec. and in vitro drug release of 98.87% after 20min. The bitterness scale 0.6 confirmed
by study on human volunteers. The taste masking of the drug confirmed by FTIR, DSC study and the in vitro
release of the DRC
Key word: Oral Disintegrating Tablet, Superdisintegrants, Indion 234, Drug Resin complex.
INTRODUCTION
Hypertension is according to WHO it is the state of
body in which systolic blood pressure is 150
mmHg and diastolic blood pressure is 95 mmHg or
more. Hypertension is usually defined by the
presence of a chronic elevation of systemic arterial
pressure above a certain threshold value.[1]
However, increasing evidence indicates that the
cardiovascular (CV) risk associated with elevation
of blood pressure (BP) above approximatel y 115 ⁄
75 mm Hg arises in a log-linear fashion.
Hypertension is a progressive CV syndrome. Early
symptoms of the syndrome are often present before
BP elevation is sustained; therefore, hypertension
cannot be classified solely by discrete BP
thresholds values. Progression is strongly
associated with functional and structural cardiac
and vascular abnormalities that damage the heart,
kidneys, brain, vasculature, and other organs and
lead to premature morbidity and death also.
Decrease in BP when target organ damage is
demonstrable or the functional precursor of target
organ damage is present and still reversible
generally reduces the risk for CV disease. Calcium
channel blockers are the type of drugs which are
used to treat the elevated blood pressure. They act
by slowing the movement of the calcium ion in to
the smooth muscle of the heart and blood vessel
walls which makes comfortable for the blood
vessel to pump out the blood easily the result is that
heart dosen’t have to work hard and it lowers the
blood pressure. Calcium channel blocker have
added benefit that slowing the heart rate which can
further reduce blood pressure and reduces the chest
pain.[2,3,4]
Verapamil hydrochloride is a calcium ion influx
inhibitor (slow-channel blocker or calcium ion
antagonist) that exerts its pharmacologic effects by
modulating the influx of ionic calcium across the
cell membrane of the arterial smooth muscle.
Calcium channel blocker binding to L-type calcium
channel and reducing calcium flux. Here muscle
does not respond calcium ion signal, Relaxes
smooth muscle of heart and slow down the elevated
blood pressure. Long-acting medications are slowly
released and helpful to provide a longer lasting