Journal of Cerebral Blood Flow and Metabolism 20:15-20 2000 The International Society for Cerebral Blood Flow and Metabolism Published by Lippincott Williams & Wilkins, Inc., Philadelphia Short Communication Detection of Tumor Necrosis Factor-a mRNA Induction in Ischemic Brain Tolerance by Means of Real-Time Polymerase Chain Reaction Xinkang Wang, Xiang Li, Joseph A. Erhardt, Frank C. Barone, and Giora Z. Feuerstein Department of Cardiovascu lar Pharmacol ogy, SmithK l ine Beecham Pharmaceuticals, King of Prussia, Pennsylvania, U.S.A. mmry: A short duration of ischemia (i.e., ischemic pre conditioning) results in significant brain protection to subse quent severe ischemic insult. Because previous studies suggest that tumor necrosis factor-x (TNF-x) plays a role in both pro moting ischemic damage and neuroprotection, the present work aimed to evaluate the expression of TNF-x mRNA in an es tablished model of ischemic preconditioning using a transient 10-minute occlusion of the middle cerebral artery. Because the level of TNF-x mRNA expression in the brain was too low to be consistently detected by Northen technique, a real-time polymerase chain reaction method was applied to quantitate the absolute copy number of TNF-x transcript in rat brain after the Tumor necrosis factor a (TNF-a) is a pleitrophic cy tokine with diverse biologic activities. TNF-a is ex pressed in monocytes/macrophages as well as many other cells including glia and neurons (Akira et al., 1990; Liu et al., 1994; Munozfernandez and Fresno, 1998). Whereas normal brain tissue has little or no TNF-a ex pression, this cytokine is significantly induced ater tran sient or permanent focal cerebral ischemia (Liu et al., 1994; Wang et al., 1994; Buttini et al., 1996). In addition, TNF-a receptors are also present in the brain and may mediate neuronal and glial activation, proliferation, dif ferentiation, and survival (Munozfernandez and Fresno, Received April 21, 1999; final revision received July 23, 1999; ac cepted July 28, 1999. Address correspondence and reprint requests to Xinkang Wang, PhD, Department of Cardiovascular Sciences, Dupont Pharmaceuticals Company, Experimental Station, E400/3420B, Wilmington, DE 19880- 0400, U.S.A. Current address for X. Wang and G. . Feuerstein is Department of Cardiovascular Sciences, DuPont Pharmaceuticals Company, Wil mington, DE 19880-0400, U.S.A. Abbreviations used: Ct, threshold cycle; MCAO, occlusion of the middle cerebral artery; PCR, polymerase chain reaction; TNF-x, tumor necrosis factor-x. 15 preconditioning procedure. TNF-x mRNA was induced in the ipsilateral cortex as early as 1 hour (27 ± I copies of mRNA per microgram of tissue compared to II ± 3 copies in sham operated samples) ater preconditioning, reached a peak level at 6 hours (49 ± 10 copies of transcript, n = 4, P < 0.01), and persisted up to 2 days. These data not only demonstrate the utility of real-time polymerase chain reaction for sensitive and accurate measurement of mRNA expression in normal and in jured tissues but also suggest a potential role of TNF-x in the phenomenon of ischemic preconditioning. y r: TNF x-Ischemic tolerance-Ischemic preconditioning-Focal stroke-TaqMan-Polymerase chain reaction. 1998). Furthermore, the expression of TNFR2 was dem onstrated to be upregulated during cerebral infection (Lucas et al., 1997). Although the precise role of TNF-a in brain function and especially in stroke is not fully understood, it has been suggested that TNF-a expression in brain ischemia is detrimental to neurons because the administration of anti-TNF-a antibodies or TNF receptor linked to poly ethylene glycol (TNFbp, which binds and inhibits TNF a) significantly reduced focal cerebral ischemic injury (Dawson et al., 1996; Brone et al., 1997; Nawashiro et al., 1997a). In addition, vv administration of TNF-a into brain parenchyma produced significant inlamma tory reaction in brain capillaries including pericapillary edema and significant leukocyte accumulation (Feuer stein et al., 1994; Liu et al., 1994). TNF-a administration into the cerebroventricular space before ischemia aug ments the extent of tissue damage and neurologic deficits (Barone et al., 1997). These results are in agreement with early studies that suggested TNF-a might play a crucial role in tissue injury during disease processes when it is released from activated lymphocytes, macrophages of