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N-Acetylcysteine
Augmentation to
Tranylcypromine in
Treatment-Resistant
Major Depression
To the Editors:
T
he treatment of major depressive dis-
order (MDD) has evolved in the past
decades with the advent of selective se-
rotonin reuptake inhibitors because of
their tolerability and safety profile. Nev-
ertheless, recent evidence indicates that
only 33% of patients achieve remission with
a single agent in real-world scenarios.
1,2
Some patients fail to remit even with com-
plex combination regimens.
3
These group
of difficult-to-treat patients represent a
major challenge for clinical psychiatrists.
3
In these instances, the use of monoamine
oxidase inhibitors (MAOIs) is often nec-
essary.
4,5
However, the Sequenced Alter-
natives to Relieve Depression (STAR*D)
trial reported that only approximately 7%
of these treatment-resistant patients remit
with MAOIs.
6
Evidence to guide sub-
sequent psychopharmacological strate-
gies for patients with MDD who did not
achieve remission after a MAOI trial
derive from a few published case re-
ports.
7,8
Here, we report for the first time
the successful use of N-acetylcysteine (NAC)
augmentation in patients who did not
achieve response after a trial with the
MAOI tranylcypromine.
Several pharmacodynamic properties
of NAC anticipate putative antidepressant
properties.
9
For instance, NAC is a pre-
cursor of glutathione, a main antioxidant
of the brain.
9
Several other actions of NAC
may be relevant to its possible antide-
pressant activity: (1) its anti-inflammatory
effects; (2) the indirect decrement of syn-
aptic release of glutamate, and (3) the fa-
cilitation of striatal dopamine release.
9
N-acetylcysteine has antidepressant prop-
erties in the rat bulbectomy model of
depression.
10
Moreover, preliminary evi-
dence indicates that adjunctive NAC may
be effective for the treatment of depres-
sive episodes of bipolar disorder.
11,12
CASE 1
In January 2011, a 22-year-old male
medical student presented with a se-
vere, treatment-refractory, first episode of
MDD without psychotic symptoms. He
presented with atypical features (rejection
sensitivity, increased appetite, hypersom-
nia, and mood reactivity) along with sui-
cidal thoughts, intention, and plans. He
had never experienced manic symptoms.
The patient did not have a personality
disorder (as assessed with the Structured
Clinical Interview for the Diagnostic and
Statistical Manual of Mental Disorders,
Fourth Edition Axis II Disorders). The
episode had been lasting for approximately
18 months. A comprehensive medical ex-
amination that included laboratory exami-
nations did not reveal abnormalities. His
mother had a history of recurrent MDD.
He was previously treated with 2 SSRIs
(escitalopram, up to 30 mg/d for 12 weeks;
and paroxetine, up to 80 mg/d for
8 weeks), venlafaxine (up to 375 mg/d
for 12 weeks), and clomipramine (up to
300 mg/d for 12 weeks). The patient did
not achieve a clear treatment response.
Therefore, we augmented clomipramine
(300 mg/d) with lithium (up to 1500 mg/d;
serum levels, 1.1 mEq/L for 4 weeks) and
quetiapine (up to 300 mg/d for 2 weeks).
His score on the 17-item Hamilton De-
pression Rating Scale (HDRS-17) was 19.
Tranylcypromine was initiated at a
daily dose of 10 mg and was then titrated
to a maximum daily dose of 90 mg for
4 weeks. The patient was on tranylcy-
promine, 90 mg/d, for 12 weeks and had a
HDRS-17 score of 12 and a Clinical
Global ImpressionVImprovement (CGI-I)
score of 3 (minimally improved). Blood
pressure was monitored throughout the
treatment, and there was no alteration. No
adverse effects were reported by the pa-
tient. At this time, we had suggested bi-
lateral electroconvulsive therapy (ECT),
but the patient declined this treatment
modality.
N-acetylcysteine was started at a
daily dose of 2 g/d 2 times a day orally
(with a 12-hour interval between doses).
After 8 weeks, the HDRS-17 score was 5,
and the CGI-I score was 1 (very much
improved). The patient has been followed
up for 7 months since then and is still
in symptomatic remission; he is now re-
garded as a very good-acting intern in his
medical school.
CASE 2
In November 2010, a 43-year-old
woman presented to our clinic with
treatment-resistant MDD. She had a previ-
ous episode 12 years ago triggered by ar-
guments with her husband, which ultimately
led to a divorce; that episode was suc-
cessfully treated with fluoxetine (daily dose,
60 mg). Fluoxetine was discontinued 1 year
after recovery. The patient was asymp-
tomatic for 10 years. However, in the past
2 years, she had a second episode of
MDD. She did not have psychotic symp-
toms, but she presented with typical
melancholic features. She had lost 7 kg
(approximately 10% of her weight) and
experienced excessive guilt, early morn-
ing awakening, psychomotor retardation,
and passive suicidal thoughts (‘‘I would
be better off dead’’). Her mother had a
history of recurrent MDD, and her oldest
sister had chronic recurrent depression and
eventually committed suicide. A compre-
hensive medical evaluation did not reveal
any abnormalities. She had been treated
with several antidepressant drugs, includ-
ing 2 SSRIs (fluoxetine, up to 50 mg/d for
12 weeks; and sertraline, up to 200 mg/d
for 2 months), duloxetine (up to 120 mg/d
for 8 weeks) and imipramine (up to
250 mg/d for 28 weeks). Lithium was
added to impramine (1200 mg/d; serum
levels, 1.2 mEq/L for 20 weeks). Because
the patient did not achieve response,
olanzapine (10 mg/d for 3 months) was
added to imipramine (250 mg/d) plus lith-
ium (1200 mg/d). Her HDRS-17 score was
still 21.
She had also been treated with a
course of 14 bilateral ECT sessions over
5 weeks. Her HDRS-17 score reduced to
17 (CGI-I score, 3: minimally improved).
After this unsuccessful intervention, we
started tranylcypromine at a daily dosage
of 10 mg, which was titrated up to 60 mg/d
for 4 weeks. The patient could not tolerate
Journal of Clinical Psychopharmacology & Volume 33, Number 5, October 2013 Letters to the Editors
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