ARTHRITIS & RHEUMATISM
Vol. 62, No. 3, March 2010, pp 908–910
© 2010, American College of Rheumatology
LETTERS
DOI 10.1002/art.27310
Rituximab monotherapy, rather than rituximab plus
antiviral drugs, for initial treatment of severe
hepatitis C virus–associated mixed cryoglobulinemia
syndrome: comment on the article by Terrier et al
To the Editor:
We read with interest the recent article by Terrier et al
(1) in which the authors report on the long-term followup of
patients with severe hepatitis C virus–associated mixed cryo-
globulinemia (HCV-MC) syndrome who were treated with
rituximab, with or without concomitant antiviral therapy. In
our opinion, the relevance of the 2 key points of the article
should be better dissected.
While the reported followup data may offer support
for the efficacy and safety of long-term rituximab therapy, any
preferential use of the combination regimen in HCV-related
vasculitis, as proposed by Terrier et al, is probably premature
at this time. A combination regimen may attack the chronic
infectious and autoimmune disorder with synergistic effects
and surely deserves investigation (1,2), but adequate studies
are still needed. Since the same group has previously excluded
rituximab monotherapy in therapeutic flow-charts for MC (3),
we will focus on this issue.
The study by Terrier and colleagues was a retrospec-
tive nonrandomized study comparing rituximab monotherapy
with combination therapy (1). The patients in the 2 groups
were quite heterogeneous with regard to both previous history
and clinical involvement, and in the study, skin and articular
manifestations were a criterion for response to treatment but
not a criterion for study inclusion. Furthermore, the authors
state that one-half of the patients treated with rituximab alone
were unresponsive to previous antiviral therapies, while also
stating that rituximab alone was used for patients for whom
antiviral therapy was contraindicated or in whom tolerance to
antiviral therapy was poor. It is conceivable that patients never
treated before with antiviral therapy may better respond to
rituximab plus antiviral therapy than to rituximab alone in
larger studies.
However, this raises the main question (2) of whether
it is better to start directly with combination therapy or with
monotherapy (presumably, rituximab) in severe HCV-MC
(more data are needed for “HCV-related vasculitis,” with 3
patients in the study by Terrier et al lacking cryoglobulins [1]).
The combination regimen, even as employed by Terrier and
colleagues (i.e., with antiviral therapy started 1 month after
rituximab), does not sufficiently distinguish between the effi-
cacy and safety of the antiviral therapy versus the B cell
depletive treatment. Response to and side effects of either
therapy may occur later and should be differentiated as early as
possible, while also considering subsequent, very long-term
treatment decisions. Whether the benefits of combination
therapy outweigh the problems with differential identification
of responses/side effects in severe cases deserves further
investigation. Rituximab monotherapy alone may be similarly
effective but more convenient as initial therapy, and antiviral
therapy may be introduced later, once the efficacy and safety
of rituximab have been better evaluated. This usually takes at
least 4–6 months. (We are using antiviral therapy, in such a
sequential schedule, 6 months after rituximab.) Combination
therapy from the beginning might indeed be more convenient
in subsets of MC, but such subsets have to be defined.
Second, a small number of cases of HCV-MC that arise
are resistant to effective antiviral therapy, which can lead to
HCV RNA negativization (4), supporting the concept that
autoimmune-related events are not driven by chronic infection
in some patients (2) (Figure 1). Even in a phase of the disease
that is dependent on both the infectious trigger and down-
stream B cell hyperactivation, however, a monotherapy di-
rected at only 1 of the 2 pathogenetic components may be
sufficient and safer (2) (Figure 1).
Randomized trials and laboratory research are needed
to better clarify these issues. A multicenter, randomized,
long-term controlled trial comparing rituximab monotherapy
versus conventional treatment in patients with MC that is
either unresponsive to or with contraindications to antiviral
therapy has been recently concluded (De Vita S: personal
communication). Better recommendations for rituximab
monotherapy in MC are awaited.
Dr. De Vita has received consulting fees, speaking fess, and/or honoraria
from Roche (less than $10,000).
Salvatore De Vita, MD
Luca Quartuccio, MD
University of Udine
Udine, Italy
1. Terrier B, Saadoun D, Sene D, Sellam J, Perard L, Coppere B, et
al. Efficacy and tolerability of rituximab with or without PEGylated
interferon alfa-2b plus ribavirin in severe hepatitis C virus–related
Figure 1. Targeting hepatitis C virus (HCV), autoimmunity, or both
in mixed cryoglobulinemia syndrome. Infection and autoreactivity may
play one role in sustaining B cell autoimmunity or autoimmune disease
and a different role in B cell expansion. There may be a strong
rationale for using monotherapy against HCV or against downstream
biologic events, or for using a combination therapy, and they all may be
useful in a single case at different stages of disease.
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