Global Journal of Pharmacology 5 (1): 27-32, 2011
ISSN 1992-0075
© IDOSI Publications, 2011
Corresponding Author: Ekramul Haque , Department of Pharmacy,BRAC University, 66-Mohakhali, Dhka-1212, Bangladesh.
Tel: +8801711952286, E-mail: haque_md.ekramul@yahoo.com.
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In vitro Free Radical Scavenging and Thrombolytic
Activities of Bangladeshi Aquatic Plant Aponogeton undulatus Roxb
Nargis S. Chowdhury, M. Badrul Alam, A.S.M. Tanbirul Haque,
1 2 3
Ronok Zahan, M. Ehsanul H. Mazumder and M. Ekramul Haque
2 4 5
Department of Pharmacy, Manarat International University, Dhaka, Bangladesh
1
Department of Pharmacy, Atish Dipankar University of Science & Technology, Banani, Dhaka, Bangladesh
2
Department of Agribusiness,
3
Atish Dipankar University of Science & Technology, Banani, Dhaka, Bangladesh
Discipline of Biomedical Science, Faculty of Medicine, Cumberland Campus, University of Sydney, Australia
4
Department of Pharmacy, BRAC University, Mohakhali, Dhaka, Bangladesh
5
Abstract: Investigation with the crude methanolic extract of Aponogeton undulatus was carried out to evaluate
its possible antioxidant and thrombolysis activity. In DPPH free radical scavenging assay, the extract exhibited
potent antioxidant activity with a IC values of 2.43±1.06 μg/ml while in ascorbic acid, the value become
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2.14±0.11 μg/ml. In thrombolytic activity using in vitro clot lysis assay method, the crude methanolic extract
was found to have significant (p<0.001) thrombolytic activity at a dose of 10 mg/ml with a miximum effect
of 20.23±1.56% while the standard streptokinase showed 46.13±3.87%. The extract was also investigated for
its antibacterial and toxic potentiality using agar diffusion and Brine Shrimp lethality bioassay, respectively.
The highest antibacterial effect was shown against Bacillus cereus (zone of inhibition 12±0.65 mm) followed
by Escherichia coli (zone of inhibition 10±0.71 mm). In this bioassay the extract showed significant toxicity to
Brine Shrimp nauplii with the LC value of 2.24±0.98 μg/ml. The study clearly indicated that the extract
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possesses good antioxidant and thromolytic activity along with broad spectrum antibacterial and toxic
potentiality.
Key words: Free radical %Thrombolysis %Aponogeton undulatus %Toxicity
INTRODUCTION Cerebral venous sinus thrombosis (CVST) is a common
Free radicals cause depletion of immune system mortality [4, 5]. Heparin, an anticoagulating agent, is the
antioxidants, change in gene expression and induce first line of treatment for CVST, because of its efficacy,
abnormal proteins and contribute to more than one safety and feasibility [6]. Thrombolytic drugs like tissue
hundred disorders in humans including atherosclerosis, plasminogen activator (t-PA), urokinase, streptokinase
arthritis, ischemia and reperfusion injury of many tissues, etc. play a crucial role in the management of patients with
central nervous system injury, gastritis, cancer and AIDS CVST [7].
[1, 2]. Undoubtedly, in vivo suppression of free radicals Plants produce wide array of bioactive principles and
is important for the human body to eliminate the toxicity constitute a rich source of medicines. In many developing
induced by free radicals. For several years, many countries, traditional medicine is one of the primary health
researchers have been investigated powerful and nontoxic care systems [8, 9]. Large scale evaluation of the local
antioxidants from natural sources, especially edible or flora exploited in traditional medicine for various
medicinal plants to prevent the free radical related biological activities is therefore necessary. Isolation and
disorders in human, which replaces the synthetic characterization of the bioactive principles ultimately
compounds because of their probable carcinogenic leading to new drug development. In view of this,
activity which are harmful to the lungs and liver [3]. our attention has been focused particularly
disorder which accompanied by significant morbidity and