178 Ann. N.Y. Acad. Sci. 961: 178–182 (2002). © 2002 New York Academy of Sciences. TGF-1-Stimulated Osteoblasts Require Intracellular Calcium Signaling for Enhanced 5 Integrin Expression LEON J. NESTI, a,b E.J. CATERSON, a MARK WANG, a RICHARD CHANG, a FELIX CHAPOVSKY, a JAN B. HOEK, b AND ROCKY S. TUAN a Departments of a Orthopaedic Surgery and b Pathology, Anatomy, and Cell Biology, Thomas Jefferson University, Philadelphia, Pennsylvania 19107, USA ABSTRACT: The osteoactive factor, transforming growth factor 1 (TGF-1), influences osteoblast activity and bone function. We recently characterized a Smad-independent TGF-1-induced Ca 2+ signal in human osteoblasts (HOB) and demonstrated its importance in cell adhesion. Here, we further elucidate the role of the TGF-1 Ca 2+ signal in the mechanics of HOB adhesion. Osteo- blast interaction with fibronectin (FN) through 51 integrin is principally re- sponsible for osteoblast-substrate adhesion. Our results show that the TGF-1 intracellular Ca 2+ signal is responsible, in part, for stimulation of 5 integrin expression, but not 1 integrin or FN expression. Increased 5 integrin pro- tein and mRNA expression was seen as early as 12 h after TGF-1 treatment, but was inhibited by cotreatment with nifedipine, a Ca 2+ channel blocker. TGF-1 increased both FN and 1 integrin protein production within 48 h, in- dependent of nifedipine cotreatment. Immunofluorescence observations re- vealed that TGF-1 increased 5 integrin staining, clustering, and colocalization with the actin cytoskeleton, effects that were blocked by nife- dipine. The TGF-1 Ca 2+ signal, a pathway crucial for HOB adhesion, en- hances 5 integrin expression, focal contact formation, and cytoskeleton reorganization. These early events are necessary for osteoblast adhesion; thus they determine the fate of the cell and ultimately affect bone function. KEYWORDS: TGF-signaling; orthopedic tissue engineering INTRODUCTION Substantial information is available indicating that the osteoactive factor, trans- forming growth factor-β1 (TGF-β1), which is crucial for bone growth and develop- ment, influences osteoblast adhesion, proliferation, differentiation, and maturation. These properties are important in considering TGF-β1 for orthopedic tissue engi- neering applications such as fracture repair, implant fixation, and structural defects. The direct effect of TGF-β1 on osteoblast activity has been well documented; how- ever, little is known about the mechanisms through which TGF-β1 exerts these ef- Address for correspondence: Leon J. Nesti, Department of Orthopaedic Surgery, Thomas Jef- ferson University, 501 Curtis Building, 1015 Walnut Street, Philadelphia, PA 19107. Voice: 215- 955-4321; fax: 215-955-4317. leonnesti@yahoo.com