Supramolecular Helical Mesomorphic Polymers. Chiral
Induction through H-Bonding
Joaquı ´n Barbera ´ , Laura Puig, Pilar Romero, Jose ´ Luis Serrano, and Teresa Sierra*
Contribution from the Instituto de Ciencia de Materiales de Arago ´ n, Consejo Superior de
InVestigaciones Cientı ´ficas, and Quı ´mica Orga ´ nica, Facultad de Ciencias, UniVersidad de
Zaragoza, 50009 Zaragoza, Spain
Received June 8, 2004; E-mail: tsierra@unizar.es
Abstract: The work described here concerns a challenge of general interest in supramolecular chemistry:
the achievement of chiral helical organizations with controlled structures. This work provides a strategy to
obtain supramolecular polymers in which a chiral helical conformation has been induced by a noncovalent
association, that is, through hydrogen bonding. Polycatenar 2,4,6-triarylamino-1,3,5-triazines, which organize
into columnar mesophases and are susceptible to H-bonding interactions, were chosen as a starting point
to build up the chiral supramolecular structure. The stacking of these mesogens has been forced to wind
in a helical way by means of H-bond association with (R)-3-methyladipic acid, within the mesophase. The
optically active columnar organization has been studied in depth by optical microscopy, differential scanning
calorimetry (DSC), X-ray diffraction, and circular dichroism. Formation of stable complexes between the
triazine units and (R)-3-methyladipic acid has also been investigated by means of NMR diffusion-ordered
spectroscopy (DOSY) experiments in chloroform.
Introduction
The significant role of helical organizations in nature [e.g.,
R-helical proteins, nucleic acids, tobacco mosaic virus (TMV)]
has stimulated the curiosity of researchers in materials chemistry.
As an example, the structure of TMV (in which the self-
assembly of 2130 polypeptide units gives rise to a columnar
organization that is driven to form a helical conformation by
interaction with an RNA chain through specific and directional
H-bonding interactions)
1
has already been used as a model for
synthetic supramolecular columnar organizations prepared from
simple molecular units.
2
Furthermore, many appealing research
works aimed at building and controlling supramolecular chiral
architectures based on helical superstructures have been re-
ported.
3,4
Indeed, interesting linear optical
5
and nonlinear optical
properties,
6
electrooptical behavior,
7,8
energy transfer,
9
etc., have
been found in synthetic helical superstructures, which are often
prepared according to the principles of supramolecular chem-
istry.
10
In this respect, our research program has been devoted
to liquid crystalline organizations and the possibility of achieving
helical columnar organizations by π-π stacking of chiral
mesogenic molecules synthesized by means of metal coordina-
tion.
8,11
In the work described here, we developed a simple strategy
based on two types of noncovalent intermolecular interaction,
that is, π-π interactions and H-bonding, which enabled the
construction of a number of supramolecular liquid crystalline
assemblies.
12
Furthermore, since the first chiral helical supramo-
lecular polymer was reported by Lehn and co-workers,
13
these
types of interaction have been successfully employed as a tool
to synthesize supramolecular structures that are capable of
adopting chiral helical organizations.
14-17
Our approach consists of merging mesomorphic arrangements
based on molecular stacking, which is promoted by π-π
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Published on Web 12/04/2004
458 9 J. AM. CHEM. SOC. 2005, 127, 458-464 10.1021/ja046644e CCC: $30.25 © 2005 American Chemical Society