RRJoLS (2015) 1-8 © STM Journals 2015. All Rights Reserved Page 1
Research & Reviews: A Journal of Life Sciences
ISSN: 2249-8656(online), ISSN: 2348-9545(print)
Volume 5, Issue 3
www.stmjournals.com
Anti-Ulcer Activity of Methanolic Extract of Mucuna
Pruriens Seed on Indomethacin Induced Ulcers
in Albino Rats
Iswar Hazarika
1
*, Panner Selvam
1
, Anju Das
2
1
Department of Pharmacology, T John College of Pharmacy, Gottigere, Bannerghatta Road,
Bangalore, Karnataka, India
2
Department of Pharmacology, the Oxford College of Pharmacy, Bangalore, Karnataka, India
Abstract
The present study was intended to investigate and evaluate the antiulcer activity of the
methanol seed extract of Mucuna pruriens using indomethacin induced ulcer in albino rats
and to determine its link between oxidant or antioxidant parameter. The extract of Mucuna
pruriens was tested on indomethacin induced gastric ulcer in albino rats. The antiulcer
activity of high dose (400 mg/kg) and low dose (200 mg/kg) of ethanolic extract of Mucuna
pruriens was assessed by measuring the ulcerative area and percentage reduction of
ulcerative area, which was compared with a standard drug misoprostol. To determine the
underlying mechanism for its antiulcer activity, the oxidant/antioxidant parameters like
glutathione peroxidase (GPO), superoxide dismutase (SOD), catalase (CAT),
myeloperoxidase (MPO), malondialdehyde (MDA) and glutathione (GSH) enzyme were
measured in the gastric tissues. Pretreatment of ethanolic extract both high dose and low dose
showed significant (p<0.001) decrease in the ulcerative area as compared to the control and
was almost as effective as the standard misoprostol. In rats given ethanolic extract, all of the
investigated antioxidant parameters increased, except for catalase (CAT). Conversely, aside
from myeloperoxidase (MPO), all oxidant parameters decreased. In conclusion, the antiulcer
activity of Mucuna pruriens may be due to its antioxidant property.
Keywords: Mucuna pruriens, indomethacin induced ulcer, ulcer area, superoxide dismutase,
catalase, glutathione
*Author for Correspondence E-mail: iswarhazarika@gmail.com
INTRODUCTION
Gastric ulcer is a symptomatic gastrointestinal
disorder that affects a considerable number of
people in the world. Its development and
progression depends to some extent on the
type of the food consumed by the patient.
Studies have shown that spicy, fatty or foods
containing caffeine stimulates acid secretion in
stomach and increase the risk of ulcer
formation [1]. Pathogenesis of peptic ulcer lies
in the localized loss of gastric as well as
duodenal mucosa. It arises when the normal
mucosal defensive factors such as mucus,
mucosal blood flow, formation of bicarbonate
ions and prostaglandin E
2
are impaired or over
powered. Also by the aggressive factor
includes acid, pepsin, NSAIDs and
Helicobacter pylori [2]. Gastric ulcer resulted
from persistent erosions and damage of the
stomach wall that might become perforated
and developed into peritonitis and massive
hemorrhage as a result of inhibition in the
synthesis of mucus, bicarbonate and
prostaglandins [3].
Side effects are the major limitation of the
presently available commercial antiulcer
drugs. For example, histamine H
2
-receptor
antagonists (e.g. cimitidine) may cause
gynecomastia in men and galactorrhea in
women while proton pump inhibitors (e.g.
omeprazole and lansoprazol) can cause nausea,
abdominal pain, constipation and diarrhea. Due
to those side effects, there is a need to find
new antiulcerogenic compound with
potentially less or no side effect. Medicinal
plants have always been the main sources of
new drugs candidates for the treatment of
gastric ulcer [4].