D. KANAGAPUSHPAM, V. RAMAMURTHY AND K. VENKATESAN 1131
approximations, this approach was successful in ration-
alizing the rigid systems like coumarin derivatives
(Murthy, Arjunan, Venkatesan & Ramamurthy, 1986).
We have assumed in these calculations that the overall
topography of the excited molecule is the same as in the
ground state. This clearly is not true and this assump-
tion is more serious in the present molecule than in rigid
molecules such as coumarins. In its reaction pathway
involving change in the hybridization of the reactive
atoms C(9) and C(14) from sp 2 to sp 3 with a lengthy
styrene side group at C(9), it would be expected that the
side group undergoes considerable positional changes in
the existing crystal lattice which might not be favour-
able from the intermolecular energy calculations. It
seems most likely that the available cavity volume
(Cohen, 1975) is insufficient as the molecular topology
undergoes very large changes in the course of the
reaction path from the reactant to the product.
We record our grateful thanks to Professor A. J.
Birch, FRS, Australian Academy of Sciences, for
suggesting this problem and Professor V. Ramakrish-
nan for useful discussions.
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Acta Cryst. (1987). C43, 1131-1134
Structure of 5-(p-Aminobenzenesulfonamido)-l-phenylpyrazole (Sulfaphenazole)*
BY H. C. PATEL AND T. P. SINGH
Department of Biophysics, All-India Institute of Medical Sciences, New Delhi - 110029, India
(Received 25 August 1986; accepted 12 January 1987)
Abstract. C~sH14N402S, Mr=314.4, monoclinic, P21/n,
a = 14.760 (3), b = 11.253 (2), c= 19.213 (4) A,
fl=109.90(3) ° , V=3001(1)A 3, Z=8, Dm=
1.397 (5), D x = 1.3916 (5) Mg m -3, 2(Mo Ktx) =
0.71069A, p=0.216mm -l, F(000)=1312, T=
293 K, final R = 0.067 for 3208 observed reflections.
The two crystallographically independent molecules A
and B in the structure have similar molecular dimen-
sions but their conformations are substantially different.
*Chemical Abstracts name: 4-amino-N-(1-phenyl-lH-pyrazol-
5-yl)benzenesulfonamide.
0108-2701/87/061131-04501.50
The six-membered benzene-ring planes in molecule
A and in molecule B are inclined to the planar pyrazole
rings at 53.5 (4) and 46.9 (4)°; 75.9 (3) and 69.1 (4) °
respectively. The two benzene-ring planes in molecule A
are mutually inclined at 12.8 (3) ° while those in
molecule B are oriented at 36.5 (4) °. Both molecules
show gauche conformations about the S--N bonds with
torsion angles of-73.7 (8) and 94.0 (8) ° respectively.
The molecules are packed in the form of hydrogen-
bonded helices which are interconnected by hydrogen
bonds and van der Waals forces through the amino N
atoms and the sulfonyl O atoms.
© 1987 International Union of Crystallography