Communication
Macromolecular
Rapid Communications
Macromol. Rapid Commun. 2012, 33, 152−157
© 2012 WILEY-VCH Verlag GmbH & Co. KGaA, Weinheim wileyonlinelibrary.com 152 DOI: 10.1002/marc.201100590
1. Introduction
Nitroxide-mediated polymerization (NMP) has experi-
enced fast development in several directions: preparation
of new and more efficient initiators,
[1–4]
kinetic investi-
gations,
[5–8]
preparation of new materials,
[9–11]
and new
applications.
[3,11,12]
The kinetic process can be grossly
described as displayed in Scheme 1.
[7]
It mainly relies on
the equilibrium between the alkoxyamine C—ON bond
homolysis ( k
d
of the dormant species) that leads to the
alkyl and nitroxyl radicals and their fast recombination
( k
c
), which maintains the self-termination reactions ( k
t
)
at very low level allowing the propagation of the poly-
meric species ( k
p
). Although NMP is efficient for most
of activated monosubstituted monomers, the NMP of
1,1-disubstituted monomers such as methyl methacrylate
is still a challenge to perform. Furthermore, in several
cases, the same alkoxyamine is not suitable for the copo-
lymerization of different monomers, or when one shifts
from bulk polymerization to either polymerization of
hydrophylic monomers or polymerization in an aqueous
medium. One way to overcome these drawbacks would
be to develop new readily tunable alkoxyamines. We
have recently reported that protonation of the nitroxyl
fragment decreases k
d
as a function of the pH,
[13]
and that
protonation of the alkyl fragment in an organic solvent
increases k
d
.
[14]
Hereafter, we present the pH dependence
of the k
d
of 1 (Scheme 2), density functional theory (DFT)
calculations unveiling the effects involved in the increase
in k
d
, and applications to NMP of styrene and sodium sty-
rene sulfonate.
In recent work, a 15-fold increase in the C–ON bond homolysis rate constant k
d
of
4-pyridylethyl-SG1-based alkoxyamine was observed upon protonation of the pyridyl moiety
in organic solvent. In this report, the pH dependence of k
d
(p K
a
= 4.7) is investigated in D
2
O/CD
3
OD (v/v 1:1). A 64-fold
increase in k
d
is observed at acidic pH. Calculations show that
the increase in k
d
upon protonation is due to both an increase
in the stabilization of the protonated 4-pyridylethyl radical
and an increase of the destabilization of the starting materials
through an increase in the polarity of the alkyl fragment. This
new alkoxyamine is applied to NMP of styrene and sodium
styrene sulfonate.
Chemically Triggered C–ON Bond Homolysis
in Alkoxyamines. Part 2: DFT Investigation and
Application of the pH Effect on NMP
Elena Bagryanskaya, Paul Brémond, Mariya Edeleva, Sylvain R. A. Marque,*
Dmitriy Parkhomenko, Valérie Roubaud, Didier Siri
0 500 1000 1500 2000 2500 3000 3500 4000
-4.0
-3.5
-3.0
-2.5
-2.0
-1.5
-1.0
-0.5
0.0
k
d
=1.6 10
-2
s
-1
ln(C/C
0
)
time (s)
k
d
=2.5 10
-4
s
-1
N
P(O)(OEt)2
O
N
*
*
1
N
P(O)(OEt)2
O
N D, Cl
1H+
H
Prof. E. Bagryanskaya, Dr. M. Edeleva, D. Parkhomenko
International Tomography Center, Institutskaya 3A, 630090
Novosibirsk, Russia
Dr. P. Brémond, Prof. S. R. A. Marque, Dr. V. Roubaud, Prof. D. Siri
Aix-Marseille Université, case 521, Avenue Escadrille
Normandie-Niemen, 13397 Marseille cedex 20, France
E-mail: sylvain.marque@univ-provence.fr Scheme 1 . Simplified scheme of NMP.
k
t
M
n+1
O N
RM
n + N O
+ M
k
d
k
c
self termination products
dormant species active species
k
p