ISSN No:2321 – 8630, V – 2, I – 1, 2015
Journal Club for Pharmaceutical Sciences (JCPS)
Manuscript No: JCPS/RES/2015/28, Received On: 22/02/2015 , Accepted On : 24/02/2015, Published On: 19/04/2015
RESEARCH ARTICLE
© All Rights Reserved by “Journals Club & Co.” 1
Development & Evaluation of Satranidazole Nano Particulate
Mucoadhesive System for Periodontitis
Urooj A. Khan
1
, Usama Ahmad
2
, M. Usama Ashhar
1
, Md. Noushad Javed
1
, Gaurav K.
Jain
1*
, Farhan J. Ahmad
1
1
Department of Pharmaceutics, Faculty of Pharmacy, Jamia Hamdard, New Delhi-110062, India
2
Nanopharmaceutical & Drug Delivery Research Lab, Faculty of Pharmacy, Integral University,
Lucknow-226026, India
ABSTRACT
Emergence of nanotechnology in medicine has revolutionized the pharmaceutical industry.It has
already cleared many hurdles associated with various delivery systems such as conventional methods,
microspheres and other microparticulate systems. Recent development in nano drug delivery systems
has proved to be efficacious in the therapeutic management strategies for dental disorders. The
effective treatment for periodontal disease has been limited due to inability of earlier formulations to
remain intact at the site of action, thereby reducing the duration of action. In this research work an
attempt has been taken to develop a mucoadhesive nano particulate system of Satranidazole (SZ), a
potent antimicrobial agent effective against various micro-organisms in dental disorders. Effect of two
preparation methods for polymeric nanoparticles have been investigated to analyze their role on mean
particle size (MPS), polydispersity index (PI), zeta potential and encapsulation efficiency (EE).
Influence of solvent system, stabilizer and polymer concentration were optimized for developing a
robust formulation. The prepared nanoparticles were coated with a mucoadhesive polymer to provide
a prolonged retention at desired site, thereby increasing the duration of action. The results indicate
that uncoated satranidazole nanoparticles exhibited smaller particle size & higher encapsulation
efficiency as compared to coated nanoparticles, however, results of in-vitro release indicate that
coated nanoparticles had much better release profiles as compared to uncoated nanoparticles.
KEYWORDS
Satranidazole, Nano Particulate System, Periodontal Disease, Mucoadhesion
INTRODUCTION
Periodontal disease is a collective term
ascribed to a number of pathological
conditions characterized by degeneration
and inflammation of gums, periodontal
ligaments, alveolar bone and dental
cementum
(1)
. Treatment method includes
use of chewable delivery systems such as
*Address for Correspondence:
Gaurav K. Jain,
Department of Pharmaceutics, Faculty of
Pharmacy, Jamia Hamdard, New Delhi-110062,
India.
Email: drgkjain@gmail.com