Research Article
Inhibitory Effect of Plant Manilkara subsericea against
Biological Activities of Lachesis muta Snake Venom
Eduardo Coriolano De Oliveira,
1
Caio Pinho Fernandes,
2,3
Eladio Flores Sanchez,
4
Leandro Rocha,
2,3
and André Lopes Fuly
1
1
Laborat´ orio de Venenos e Toxinas de Animais e Avaliac ¸˜ ao de Inibidores, Departamento de Biologia Celular e Molecular,
Instituto de Biologia, Universidade Federal Fluminense, Outeiro de S˜ ao Jo˜ ao Batista, 3º andar, Sala 310, 24020-141 Niter´ oi, RJ, Brazil
2
Programa de P´ os-Graduac ¸˜ ao em Ciˆ encias Aplicadas a Produtos para a Sa´ ude, Faculdade de Farm´ acia,
Universidade Federal Fluminense, 24220-900 Niter´ oi, RJ, Brazil
3
Programa de P´ os-Graduac ¸˜ ao em Biotecnologia Vegetal, Centro de Ciˆ encias da Sa´ ude, Universidade Federal do Rio de Janeiro,
21941-599 Rio de Janeiro, RJ, Brazil
4
Centro de Pesquisa e Desenvolvimento, Fundac ¸˜ ao Ezequiel Dias, 30510-010 Belo Horizonte, MG, Brazil
Correspondence should be addressed to Andr´ e Lopes Fuly; andfuly@vm.uf.br
Received 28 August 2013; Revised 9 December 2013; Accepted 10 December 2013; Published 8 January 2014
Academic Editor: Leonardo A. Calderon
Copyright © 2014 Eduardo Coriolano De Oliveira et al. his is an open access article distributed under the Creative Commons
Attribution License, which permits unrestricted use, distribution, and reproduction in any medium, provided the original work is
properly cited.
Snake venom is composed of a mixture of substances that caused in victims a variety of pathophysiological efects. Besides
antivenom, literature has described plants able to inhibit injuries and lethal activities induced by snake venoms. his work describes
the inhibitory potential of ethanol, hexane, ethyl acetate, or dichloromethane extracts and fractions from stem and leaves of
Manilkara subsericea against in vivo (hemorrhagic and edema) and in vitro (clotting, hemolysis, and proteolysis) activities caused
by Lachesis muta venom. All the tested activities were totally or at least partially reduced by M. subsericea. However, when L. muta
venom was injected into mice 15 min irst or ater the materials, hemorrhage and edema were not inhibited. hus, M. subsericea
could be used as antivenom in snakebites of L. muta. And, this work also highlights Brazilian lora as a rich source of molecules
with antivenom properties.
1. Introduction
Snakebites are a public health problem that afects mainly
poor people who live in rural areas of Africa, Asia, Latin
America, and Oceania [1, 2]. According to World Health
Organization, it is estimated that up to ive million people are
bitten by snakes every year, and of these, 100,000 deaths occur
annually, with 400,000 amputations and other severe health
consequences (such as infection, tetanus, and scarring). Poor
access to health care and scarcity of antivenoms increase the
severity of the injuries and their outcomes. Snake venoms
are a complex mixture of proteins, including metallopro-
teinase, serine protease, phospholipase A
2
, disintegrins, C-
type lectins, myotoxins, and others [3, 4]. Lachesis muta
(Bushmaster) is the longest venomous snake in the Americas
and is distributed in the equatorial forests east of the Andes,
ranging from eastern Ecuador, Colombia, Peru, northern
Bolivia, and eastern and northern Venezuela, to Guyana,
French Guyana, Surinam, and northern Brazil. Within their
range, they are oten abundant and are an important cause of
snakebites [5]. L. muta snakebites are mainly characterized by
systemic (generalized bleeding, coagulopathy, renal failure,
and shock) and local efects (pain, hemorrhage, edema, and
necrosis) [6, 7]. In South America, B. jararaca has a higher
incidence of accidents (95%) than L. muta (2%), but, on the
other hand, L. muta bites led to more severe symptoms (listed
above) and have lethality indexes three times higher than B.
jararaca [8]. hus, reducing these indexes is necessary and
must be fast.
Although antivenoms are efective against systemic efe-
cts, they do not inhibit the local efects. And, a few countries
produce antivenom of adequate quality as well. Moreover,
Hindawi Publishing Corporation
BioMed Research International
Volume 2014, Article ID 408068, 7 pages
http://dx.doi.org/10.1155/2014/408068