Hindawi Publishing Corporation
Clinical and Developmental Immunology
Volume 2013, Article ID 679804, 8 pages
http://dx.doi.org/10.1155/2013/679804
Research Article
Trichostatin A Promotes the Generation and Suppressive
Functions of Regulatory T Cells
Cristian Doñas,
1,2
Macarena Fritz,
1,2
Valeria Manríquez,
3
Gabriela Tejón,
3
María Rosa Bono,
3
Alejandra Loyola,
2,4
and Mario Rosemblatt
1,2,3
1
Departamento de Ciencias Biol´ ogicas, Universidad Andr´ es Bello, Rep´ ublica 275, Santiago, Chile
2
Fundaci´ on Ciencia & Vida, Avenida Za˜ nartu 1482,
˜
Nu˜ noa, Santiago, Chile
3
Laboratorio de Inmunolog´ ıa, Departamento de Biolog´ ıa, Facultad de Ciencias, Las Palmeras 3425,
˜
Nu˜ noa,
Universidad de Chile, Santiago, Chile
4
Universidad San Sebasti´ an, Avenida Lota 2465, Providencia, Santiago, Chile
Correspondence should be addressed to Mario Rosemblatt; mrosemblatt@cienciavida.cl
Received 30 January 2013; Revised 9 April 2013; Accepted 9 April 2013
Academic Editor: Nicolaus Kroger
Copyright © 2013 Cristian Do˜ nas et al. his is an open access article distributed under the Creative Commons Attribution License,
which permits unrestricted use, distribution, and reproduction in any medium, provided the original work is properly cited.
Regulatory T cells are a speciic subset of lymphocytes that suppress immune responses and play a crucial role in the maintenance
of self-tolerance. hey can be generated in the thymus as well as in the periphery through diferentiation of na¨ ıve CD4
+
T cells.
he forkhead box P3 transcription factor (Foxp3) is a crucial molecule regulating the generation and function of Tregs. Here we
show that the foxp3 gene promoter becomes hyperacetylated in in vitro diferentiated Tregs compared to na¨ ıve CD4
+
T cells. We
also show that the histone deacetylase inhibitor TSA stimulated the in vitro diferentiation of na¨ ıve CD4
+
T cells into Tregs and
that this induction was accompanied by a global increase in histone H3 acetylation. Importantly, we also demonstrated that Tregs
generated in the presence of TSA have phenotypical and functional diferences from the Tregs generated in the absence of TSA. hus,
TSA-generated Tregs showed increased suppressive activities, which could potentially be explained by a mechanism involving the
ectonucleotidases CD39 and CD73. Our data show that TSA could potentially be used to enhance the diferentiation and suppressive
function of CD4
+
Foxp3
+
Treg cells.
1. Introduction
Regulatory T cells (Treg) are a speciic subset of lymphocytes
that suppress immune responses and play a crucial role in
the maintenance of self-tolerance [1, 2]. heir development
and function are programmed by the forkhead box P3
transcription factor Foxp3, which is predominantly expressed
in CD4
+
CD25
+
Treg cells [1, 3]. Tregs actively suppress the
activation and expansion of autoreactive immune cells to
limit the duration and extent of inlammation. herefore,
a decrease in Treg activity can contribute to autoimmunity
and inlammatory diseases [4]. Because of their suppressive
capacities, Tregs represent a promising strategy for inducing
tolerance to self- and non-self-antigens in such diseases.
In recent years, increasing evidence has demonstrated
the role of epigenetic alterations in the etiology of many
autoimmune and inlammatory diseases through changes in
DNA methylation and histone modiications [5, 6]. herefore,
it is important to determine crucial histone modiications for
Treg development and function and to study compounds able
to revert or modify epigenetic patterns.
Among histones modiications is acetylation, which
occurs at lysine residues mainly on their amino-terminal tails.
his posttranslational modiication is dynamic and its overall
efect on gene expression depends on the balance between
histone acetyltransferases (HATs) and histone deacetylases
(HDACs) [7, 8]. HDACs typically dampen histone-DNA and
histone-non histone protein interactions [9, 10], but they also
regulate the function of non-histone proteins [11].
Histone deacetylase inhibitors (HDACi) such as tricho-
statin A (TSA) are small molecule compounds capable of
inhibiting class I, II, and IV HDAC families of enzymes [12].