IJSRSET184485 | Received : 05 March | Accepted : 16 March 2018 | March-April-2018 [(4) 4 : 300-303 ]
© 2018 IJSRSET | Volume 4 | Issue 4 | Print ISSN: 2395-1990 | Online ISSN : 2394-4099
Themed Section : Engineering and Technology
300
Drug Profile of Emtricitabine and Tenofovir AF
N. MD. Akram
1
, Dr. M. Umamahesh
2
1
Research Scholar, Department of Chemistry, Rayalaseema University, Kurnool, Andhra Pradesh, India
2
Professor & HOD of chemistry, Rajeev Gandhi Memorial College of Engineering & Technology (RGMCET),
Nandyal, Kurnool (Dt). Andhra Pradesh, India
ABSTRACT
Emtricitabine and Tenofovir alafenamide (tenofovir AF) is a novel oral prodrug of the nucleos(t)ide reverse
transcriptase inhibitor (NRTI) tenofovir that has several pharmacological advantages over tenofovir disoproxil
fumarate (tenofovir DF), including increased plasma stability and reduced tenofovir systemic exposure.
Tenofovir AF has been coformulated with emtricitabine for the treatment of adults and adolescents with HIV-1
infection.
Keywords: Emtricitabine, Tenofovir alafenamide, NRTI.
I. INTRODUCTION
Drug Profile of Emtricitabine
Molecular structure
Figure 1. Structure of Emtricitabine
IUPAC Name 4-amino-5-fluoro-1-[(2R,5S)-2-(hydroxymethyl)-1,3- oxathiolan-5-yl]-1,2-
dihydropyrimidin-2-one.
CAS Number 143491-57-0
Drug Bank DB00879 (APRD00226)
Molecular formula C8H10FN3O3S
Molecular weight 247.248 gm/mol
Category Antiretroviral
Description Emtricitabine is a nucleoside reverse transcriptase inhibitor for the treatment
of HIV infection in adults.