Madridge J Anal Sci Instrum.
ISSN: 2638-1532
56 Volume 3 • Issue 1 • 1000111
Madridge
Journal of Analytical Sciences and
Instrumentation
Research Article Open Access
Manipulation of Different ratio Dependent approaches
for Determination of Pravastatin in the presence of
Pioglitazone in Pharmaceutical Preparation
Nasr M. El-Abasawi, Khalid A.M. Attia, Ahmad A. M, Abo-serie and Ashraf Abdel-Fattah*
Pharmaceutical Analytical Chemistry Department, Faculty of Pharmacy, Al-Azhar University, 11751 Nasr City, Cairo, Egypt
Article Info
*Corresponding author:
Ashraf Abdel-Fattah
Pharmaceutical Analytical Chemistry
Department
Faculty of Pharmacy
Al-Azhar University
11751 Nasr City, Cairo
Egypt
Tel: +201009408060
Email: ashraf.abdelfattah@hotmail.com
Received: February 16, 2018
Accepted: March 3, 2018
Published: March 9, 2018
Citation: El-Abasawi NM, Attia KAM,
Aboserie AAM, Morshedy S, Abdel-Fattah A.
Manipulation of Different ratio Dependent
approaches for Determination of Pravastatin in
the presence of Pioglitazone in Pharmaceutical
Preparation. Madridge J Anal Sci Instrum.
2018; 3(1): 56-61.
doi: 10.18689/mjai-1000111
Copyright: © 2018 The Author(s). This work
is licensed under a Creative Commons
Attribution 4.0 International License, which
permits unrestricted use, distribution, and
reproduction in any medium, provided the
original work is properly cited.
Published by Madridge Publishers
Abstract
Objective: This study aimed to develop three simple UV spectrophotometric methods
for determination of pravastatin sodium in the presence of pioglitazone hydrochloride
without previous separation.
Methods: Manipulating ratio spectra were developed for the interested methods. The
first method is the ratio subtraction using 16 µg/mL of pioglitazone hydrochloride as a
divisor. The second method is an amplitude modulation using the normalized spectrum
of pioglitazone hydrochloride as a divisor (1 µg/mL) the peak amplitudes of ratio spectra
were measured at isoabsorptivity point 251.4 nm. The third method is the ratio difference
using 14 µg/mL of pioglitazone hydrochloride as a divisor, where the peak amplitudes
of ratio spectra were measured at 240 and 246.4 nm.
The results and discussion: The calibration curve is a linear over the concentration
range of 2-20 µg/mL, the proposed methods were validated according to International
Conference on Harmonization (ICH) guidelines and successfully applied for the
determination of pravastatin sodium in the presence of pioglitazone hydrochloride in
their combined pharmaceutical formulation, Pravazon® capsules with high sensitivity.
Conclusion: The proposed three methods are simple, rapid, economical, accurate and
precise for determination of pravastatin sodium in the presence of pioglitazone
hydrochloride without previous separation.
Keywords: Pravastatin Sodium; Pioglitazone Hydrochloride; Ratio Subtraction; Amplitude
Modulation; Ratio Difference.
Introduction
Pravastatin sodium (PRV), (Figure 1a), is sodium (3R,5R)-7-{(1S,2S,6S,8S,8aR)-
1,2,6,7,8,8a-hexahydro-6-hydroxy-2-methyl-8-[(S)-2-methylbutyryloxy]-1-naphthyl}-
3,5-dihydroxyheptanoate [1,2]. It is a selective and competitive inhibitor of 3-hydroxy-3-
methylglutaryl -coenzyme A (HMG-CoA) reductase, the rate-limiting enzyme that
converts HMG-CoA to mevalonate, a precursor of cholesterol [3]. PRV is a member of
the class of statins, used to treat hypercholesterolemia and related conditions and to
prevent cardiovascular disease. It increases the number of hepatic low density lipoprotein
(LDL) receptors on the cell surface to enhance uptake and catabolism of LDL. Secondly,
PRV inhibits hepatic synthesis of very low density lipoprotein (VLDL), which reduces the
total number of VLDL and LDL particles [4].
Pioglitazone hydrochloride (PGZ), (Figure. 1b), is 5-[[4-[2-(5-Ethyl-2-pyridinyl)
ethoxy]phenyl]methyl]-2,4-thiazolidinedione hydrochloride [5]. It is a thiazolidine-dione
oral antidiabetic agent that improves insulin sensitivity. It is used in the treatment of
ISSN: 2638-1532