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The Pharma Innovation Journal 2021; 10(5): 240-243
ISSN (E): 2277- 7695
ISSN (P): 2349-8242
NAAS Rating: 5.23
TPI 2021; 10(5): 240-243
© 2021 TPI
www.thepharmajournal.com
Received: 03-03-2021
Accepted: 23-04-2021
Shruti
Department of Biochemistry,
College of Basic Sciences and
Humanities, G. B. Pant
University of Agriculture and
Technology, Pantnagar,
Uttarakhand, India
AH Ahmad
Department of Veterinary
Pharmacology & Toxicology,
College of Veterinary and Animal
Sciences, G. B. Pant University
of Agriculture and Technology,
Pantnagar, Uttarakhand, India
Sanjeev Agarwal
Department of Biochemistry,
College of Basic Sciences and
Humanities, G. B. Pant
University of Agriculture and
Technology, Pantnagar,
Uttarakhand, India
Ashutosh Dubey
Department of Biochemistry,
College of Basic Sciences and
Humanities, G. B. Pant
University of Agriculture and
Technology, Pantnagar,
Uttarakhand, India
AK Verma
Department of Biochemistry,
College of Basic Sciences and
Humanities, G. B. Pant
University of Agriculture and
Technology, Pantnagar,
Uttarakhand, India
Corresponding Author:
AK Verma
Department of Biochemistry,
College of Basic Sciences and
Humanities, G. B. Pant
University of Agriculture and
Technology, Pantnagar,
Uttarakhand, India
Evaluation of in vitro anti-inflammatory activity in
Berberis lyceum Royle of Shivalik range of Himalaya
Shruti, AH Ahmad, Sanjeev Agarwal, Ashutosh Dubey and AK Verma
Abstract
Berberis lyceum Royle is a traditional medicinal plant of the Shivalik range of Himalaya, India, and
reported first time in vitro anti-inflammatory potentials in the root, stem, and leaves against denaturation
of protein. The different concentration of B. lyceum Royle extract, pure berberine, and diclofenac as
standard was incubated with albumin in controlled experimental conditions and subjected to determine
the absorbance and to measure their viscosity. The assay is based on the denaturation of protein upon the
heat treatment as the anti-inflammatory agent will stabilize or prevent the protein from denaturation. A
concentration-dependent inhibition of protein (albumin) denaturation by the B. lyceum Royle and
berberine was found in both. However, hydroethanolic extract B. lyceum Royle was found to more
effective when compared to pure berberine and diclofenac. High anti-inflammatory effect of
hydroethanolic extract due to the synergistic effect of other phytoconstituents present in B. lycium extract
along with berberine. Therefore from the present study, we can conclude that both berberine and B.
lyceum Royle possess anti-inflammatory activity.
Keywords: Anti-inflammatory, Berberine lyceum Royle, diclofenac, Berberine, protein denaturation,
viscosity
Introduction
Inflammation is a pathophysiological response of the defense mechanism of the living system
which is characterized by redness, edema, fever, pain, and loss of function as a result of any
tissue damage, injury, or pathogen. This is a mechanism of defense however loss of regulatory
mechanism i.e. when the inflammation is allowed to continued and unchecks it results in auto-
immune or auto-inflammatory disorders, neurodegenerative disease, or cancer
[1]
. Steroidal
anti-inflammatory drugs (SAID) and non-steroidal anti-inflammatory drugs (NSAID) are
being used to treat acute inflammatory disease, but the success of these drugs is limited in case
of chronic inflammatory disorders such as rheumatoid arthritis, atherosclerosis, type 2
diabetes, Alzheimer’s disease, and atopic dermatitis. Also, the long-term use of these drugs
can have an adverse effect too i.e., gastric ulcers, therefore there is a need for new and safe
anti-inflammatory agents and plant-derived medicine are one of the ongoing research
candidates. The advantages of plant-based medicines are their perceived efficacy, low cost,
and less incidence of serious adverse effects
[2, 3]
.
Berberis lyceum Royle belongs to the family of Berberidaceae, often used as a traditional
medicine plant by the local people of the Himalayan region. It is an evergreen shrub
commonly named Kilmoda or Daruhaldi because of the presence of yellow color pigment i.e.
Berberine in the roots of the plant. The other chemical constituents found in B. lycium are
berbamine, chinabine, karakoramine, palmatine, sindamine etc. however the berberine is the
major bioactive compound that is mainly found in the roots of the plant, and an appreciable
amount found in the leaves, stems, and berries
[4]
It is found to be effective for eye infection,
diabetes, obesity, hemorrhoids, wound healing, dysentery, skin disease, uterine and vaginal
disorder
[5-7]
. Berberine (5,6-dihydro-9,10-dimethoxybenzo(g)-1,3-benzodioxolo(5,6-
a)quinolizinium) is an isoquionide alkaloid found in plants belong Berberidaceae family. It is
a yellow-colored powder, odorless with a characteristic alkolodial taste
[8]
. It is a relevant
molecule in pharmacology and medicinal chemistry. Berberine is now manufactured by
chemical synthesis also. For clinical purposes, the sulfate or chloride salt of berberine is
generally used. Berberine is also used for the synthesis of several bioactive derivatives by the
means of condensation, modification, and substitution of functional groups in strategic
positions for the design of new, selective, and powerful drugs
[9, 10]
. Various clinical and pre-
clinical studies on berberine clinical show the curative and protective effect against many