Print ISSN 2319-2003 | Online ISSN 2279-0780
doi: 10.5455/2319-2003.ijbcp20150225
IJBCP International Journal of Basic & Clinical Pharmacology
www.ijbcp.com International Journal of Basic & Clinical Pharmacology | January-February 2015 | Vol 4 | Issue 1 Page 139
Research Article
Evaluation of wound healing activity of topical phenytoin in an excision
wound model in rats
Sarita Mulkalwar*, Lopamudra Behera, Pravin Golande, Rahul Manjare, Harshal Patil
INTRODUCTION
Wound is defned as a disruption of cellular and anatomical
or functional continuity of living tissue.
1
Wound healing is
the process of restoration of physical integrity of internal or
external body structures and involves a complex interaction
between the cells and various other factors. The healing
process consists of a sequence of overlapping events
including inflammatory responses, regeneration of the
epidermis, shrinkage of the wound and fnally connective
tissue formation and remodelling.
2
Wound healing is a signifcant healthcare problem in today’s
medical practice. Appropriate treatment and wound care
accelerate the healing process and prevent infection and
chronicity of the wound.
2
Oral phenytoin was introduced into therapy in 1938 and
widely used for management of convulsions. On long-
term administration of phenytoin, it produces gingival
hypertrophy and by virtue of this property, studies on its
effect on wound healing were undertaken.
3
According to
few studies, phenytoin possesses wound healing activity,
but there are few contradictory studies. In view of these
conficting results, the present study was planned to evaluate
the effect of topical phenytoin on the rate of wound healing
in an excision wound model and compare with petroleum
jelly and povidone iodine.
METHODS
The present study was carried out in Dr. D. Y. Patil Medical
College, Hospital and Research Centre, Pimpri, Pune,
Maharashtra, after approval from Institutional Animal Ethics
Committee (IAEC).
Animals
A total of 32, healthy (150-200 g) Sprague-Dawley rats
of either sex, aged 12 weeks bred locally in the animal
house of our college were used. The animals were kept in
ABSTRACT
Background: Wound healing is a signifcant healthcare problem in today’s medical
practice. Despite extensive treatment modalities that are supposed to hasten the
wound healing process, the outcomes of existing methods are far from optimal. One
such agent that has been tried previously and found controversial in wound healing is
phenytoin. Therefore, this study was planned to evaluate and compare wound healing
effect of topical phenytoin with povidone iodine ointment in rats.
Methods: This study was conducted after approval from Institutional Animal Ethics
Committee (IAEC). Wound healing activity of topical phenytoin (1 g% and 2 g%)
was assessed in excision wound model in Sprague Dawley rats (n=8), which was
compared with topical petroleum jelly and povidone iodine ointment. Parameters
studied included wound area on day 0, 4, 8, 12, 16, 20, percentage wound contraction,
percentage wound healing from day 0 to day 20 and period of re-epithelisation.
Results: Wound surface area decreased in all treatment groups from day 0 through
day 20 and the percentage wound closure was better in both the preparations (1% and
2%) of phenytoin when compared wih control and povidone iodine, but this was not
statistically signifcant. Furthermore, the days required for complete re-epithelisation
were less with phenytoin treated groups. There was no statistical difference between
both the preparations of phenytoin.
Conclusion: In this study, it was found that topical phenytoin accelerates wound
healing process in an excision wound model.
Keywords: Epithelization, Phenytoin, Wound contraction
Department of Pharmacology,
Dr. D. Y. Patil Medical
College, Pimpri, Pune,
Maharashtra, India
Received: 18 December 2014
Accepted: 09 January 2015
*Correspondence to:
Dr. Sarita Mulkalwar,
Email: smulkal@hotmail.com
Copyright: © the author(s),
publisher and licensee Medip
Academy. This is an open-
access article distributed under
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Commons Attribution Non-
Commercial License, which
permits unrestricted non-
commercial use, distribution,
and reproduction in any
medium, provided the original
work is properly cited.