*Corresponding author,
e-mail : nagina17001@mail.unpad.ac.id (N. Belali)
https://doi.org/10.24198/idjp.v1i3.23491
© 2019 Belali et al
Vol 1, Issue 3, 2019 (99-104)
http://journal.unpad.ac.id/idjp
Solvent Evaporation as an Efcient Microencapsulating Technique for Taste
Masking in Fast Disintegrating Oral Tablets
Nagina G. Belali
1,2*
, Anis Y. Chaerunisaa
2
1. Department of Pharmaceutics, Faculty of Pharmacy, University of Kabul - Afganistan
2. Department of Pharmaceutics, Faculty of Pharmacy, Universitas Padjadjaran, Sumedang 45363,
Indonesia
Received: 4 Sep 2019/Revised: 30 Sep 2019/Accepted: 30 Sep 2019/Published: 1 Oct 2019
ABSTRACT
Microencapsulation is an extensively used technology of present era, that has been applied to various
felds like pharmaceutical industry, agriculture, cosmetics and food technology. With the help of which
liquid or solid material can be encapsulated inside a polymeric coating flm for various reasons such
as taste masking, control release and enhancing stability and etc. Microencapsulation can be achieved
with diferent approaches and methods but one of the popular and frequently used feasible method is
Solvent evaporation. Solvent evaporation is based on emulsifcation, solvent evaporation and extraction
of microspheres, recently many variations have been made in this technology to improve the yield and
properties of microspheres. Solvent evaporation has been widely used in microencapsulating for diferent
purposes one of which is taste masking of bitter drugs in fast disintegrating oral tablets, for pediatric
and geriatric use. FDTs are center of attraction due to their merits and feasibility of use for people with
problem of dysphagia at the same time, it can also improve bioavailability and time of action of drugs.
The main focus of current review is use of solvent evaporation technique for taste masking of bitter
drugs in production of fast disintegrating oral tablets. In this review, we will summarize uses, novelties
and variations in Solvent Evaporation technique, preparation technique, materials used, merits and
demerits of this method over other microencapsulation method in taste masking.
Keywords: Microencapsulation, Solvent Evaporation, FDTs, extraction, microspheres
1. Introduction
In last decade many novelties and development
has been shown up in feld of pharmaceutics, one of
which is encapsulation of drugs that can be done on
nano and micro scale. However, Microencapsulation
is a technique that has been used for several decades,
it’s a term that present microspheres with a size of
1µm or less, liquid or solid particles encapsulated
with a secure external layer that ofers merits such
as control drug release, better drug efcacy, better
bioavailability, better drug stability, and low toxicity.
[1] Till now diferent techniques have been used for
microencapsulation such as solvent evaporation,
spray drying, polymerization, coacervation, and
phase separation and most of them have been applied
in production of fast disintegrating oral tablets, [2]
for example oxalic acid was microencapsulated
by coacervation method [3] also metformin
hydrochloride was microencapsulated with same
approach of coacervation as sited in [4], taste masked
ofoxacin microspheres by solvent evaporation,[5]
microencapsulation of antioxidant compounds from
black berry [6] microencapsulation of carotenoids
[7], moreover taste masked microspheres of
famotidine that were applied in preparation of
famotidine orally disintegrating tablets, reported by
Jiachen Xu [8] were also prepared by spray drying
approach, trioctylmethylammonium chloride
(TOMAC) microencapsulation was reported to be
performed by suspension polymerization technique
as narrated by [9].
2. Solvent evaporation technique
Solvent evaporation is a frequently used in
fabrication of micro and nanoparticles, moreover it
has been used in fabrication of hydrophobic lipid