Silva‑Pinto et al. Malar J (2017) 16:43
DOI 10.1186/s12936‑017‑1698‑y
RESEARCH
Artemether‑lumefantrine and liver
enzyme abnormalities in non‑severe
Plasmodium falciparum malaria in returned
travellers: a retrospective comparative study
with quinine‑doxycycline in a Portuguese
centre
André Silva-Pinto
*
, Rogério Ruas, Francisco Almeida, Raquel Duro, André Silva, Cândida Abreu
and António Sarmento
Abstract
Background: Artemisinin-based therapy is the current standard treatment for non-severe malaria due to Plasmo-
dium falciparum. The potential for asymptomatic liver toxicity of this therapy and its implication in clinical practice is
currently unknown. The aim of this study is to assess the hepatic function in patients treated with a standard three-
day artemisinin-based regimen and to compare it with the quinine-doxycycline regimen.
Methods: Retrospective and comparative study of returned adult travellers admitted with non-severe P. falciparum
malaria. Fifty-seven patients were included: 19 treated with artemisinin-based therapy and 38 with quinine-doxycy-
cline therapy.
Results: During treatment, when compared with quinine-doxycycline group, the artemisinin-lumefantrine group
presented a higher proportion of significant liver enzyme abnormalities (42 vs. 5%, p < 0.01) and a higher peak value
of aspartate aminotransferase (131 vs. 64 U/L, p < 0.01) and alanine aminotransferase (99 vs. 75 U/L, p = 0.05). None of
the patients was symptomatic, there were no treatment interruptions and all patients achieved clinical cure.
Conclusions: Treatment of uncomplicated falciparum malaria with artemisinin-based therapy might cause asympto-
matic liver enzyme abnormalities in the first days of treatment. Nevertheless, these liver enzyme abnormalities seem
to be harmless, asymptomatic and self-limited.
Keywords: Malaria, Artemether–lumefantrine, Liver dysfunction, Plasmodium falciparum
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Background
Artemisinin based combination therapy (ACT) is the
current standard treatment for uncomplicated malaria
caused by Plasmodium falciparum [1]. Owing to their
rapid onset of action and quick elimination, artemisinin
derivatives are very efective in reducing parasite load
and have favourable safety and tolerability profles [2, 3].
In Portugal, artemether/lumefantrine fxed dose combi-
nation (AL), currently the only available ACT, came into
medical use in 2013 and is an alternative to quinine plus
doxycycline (QD), the previous frst-line regimen [1]. Te
main reasons for this paradigm change are the safety and
tolerability profles of AL and the remaining ACT regi-
mens compared to QD [3, 4].
Open Access
Malaria Journal
*Correspondence: pintoandre@gmail.com
Infectious Diseases Department, Centro Hospitalar São João, Alameda
Professor Hernani Monteiro, 4200 Porto, Portugal