1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24 25 26 27 28 29 30 31 32 33 34 35 36 37 38 39 40 41 42 43 44 45 46 47 48 49 50 51 52 53 54 55 56 57 58 59 60 61 62 63 64 65 66 67 68 69 70 71 72 73 74 75 76 77 78 79 80 81 82 83 84 85 86 87 88 89 90 91 92 93 94 95 96 97 98 99 100 101 102 103 104 105 106 107 108 109 110 111 112 ORIGINAL INVESTIGATION Decreased whole-blood global DNA methylation is related to serum hormones in anorexia nervosa adolescents L. TREMOLIZZO 1 * , E. CONTI 1 * , M. BOMBA 2 , O. UCCELLINI 2 , M.S. ROSSI 2 , M. MARFONE 2 , F. CORBETTA 2 , M.E. SANTARONE 1 , M.E. RAGGI 3 , F. NERI 2 , C. FERRARESE 1 & R. NACINOVICH 2 1 Department of Neurology, 2 Department of Child Neuropsychiatry, San Gerardo Hospital, Monza and University of Milano-Bicocca, Monza, Italy, and 3 Clinical Analysis Laboratory, “Eugenio Medea” Scientific Institute, Bosisio Parini (LC), Italy Abstract Objectives. The one-carbon metabolism, also known as methionine-homocysteine cycle, governs the dynamics of DNA methylation, epigenetically regulating gene expression, and has been reported altered in anorexia nervosa (AN) adult patients. The aim of this study consisted in assessing whole-blood DNA methylation in adolescent AN patients, assessing its significance in relationship to clinical and hormonal variables. Methods. Whole-blood global DNA methylation was measured as incorporation of [ 3 H]dCTP following HpaII cut in 32 adolescent females affected by restrictive type AN and compared to 13 healthy controls. Homocysteine, vitamin B 12 and folate plasma levels were assessed as well as fasting plasma levels of leptin and steroid hormones. Clinical variables, including severity and associate states and traits, were assessed by means of the EDI-3, CDI and STAI-Y scales. Results. We confirm that whole-blood global DNA methylation is modestly albeit significantly reduced in AN adolescents with respect to controls, correlating with plasma leptin and steroid hormone levels. Conversely, clinical traits did not correlate with the outcome variable. Conclusions. A better definition of the epigenetic dysregulation underlying AN pathology or vulnerability might lead to develop useful markers for diagnosis, prognostic classification and tailored therapeutic interventions in these vulnerable patients since the earliest phases of their disease. Key words: anorexia nervosa, DNA methylation, whole blood, biomarkers, epigenetics Introduction Anorexia nervosa (AN) is a complex neuropsychiat- ric eating disorder strictly associated to brain circuit dysfunctions that still need to be fully elucidated (Hay and Sachdev 2011). This disrupted neurocir- cuitry in AN conceivably underlies major synaptic rearrangements during adolescence or pre-adolescence, a critical period for the maturing brain, when pivotal changes take place driven by hormonal, physical and socio-environmental strictly intertwined forces (Krassas 2003; Blakemore et al. 2010). Epigenetic modifications of DNA and chromatin histones clearly represent one major brain function determinant at the interface of the gene–environment interaction both during the ontogenesis and in adulthood, as previously shown in the setting of other neuropsychi- atric conditions and treatments (Tremolizzo et al. 2002, 2013a; Weaver et al. 2004). Among environ- mental modifiers of the epigenoma, diet certainly plays a major role, further strengthening the link with cancer, the prototypical epigenetic disease among other complex disorders (Parle-McDermott and Ozaki 2011; Kaelin and McKnight 2013). Specifically, maternal diet has been repeatedly shown in animal models to influence the epigenetic pattern in the offspring (Waterland et al. 2006), determining various adult phenotypes of disease (Sinclair et al. 2007). Human studies also have shown demethyla- tion at the imprinted insulin-like growth factor 2 ( IGF2) locus associated to higher fat density and * These authors equally contributed to the work. Correspondence: Lucio Tremolizzo, MD, PhD, Section of Neurology, DCMT, University of Milano-Bicocca, S. Gerardo Hospital, via Pergolesi 33, 20900 Monza (MI), Italy. Tel: 39 2 6448 8128. Fax: 39 2 6448 8108. E-mail: lucio.tremolizzo@unimib.it (Received 22 July 2013; accepted 21 October 2013) The World Journal of Biological Psychiatry, 2013; Early Online: 1–7 ISSN 1562-2975 print/ISSN 1814-1412 online © 2013 Informa Healthcare DOI: 10.3109/15622975.2013.860467