Carbohydrate Research 337 (2002) 851 – 861 www.elsevier.com/locate/carres The crystal structure of the -cellobiose·2 NaI·2 H 2 O complex in the context of related structures and conformational analysis Zenaida Peralta-Inga, a Glenn P. Johnson, b Michael K. Dowd, b Jacob A. Rendleman, c Edwin D. Stevens, a, * Alfred D. French b, * a Department of Chemistry, Uniersity of New Orleans, New Orleans, LA 70148, USA b US Department of Agriculture, Southern Regional Research Center, 1100 Robert E. Lee Bouleard, New Orleans, LA 70124, USA c National Center for Agricultural Utilization Research, 1815 N Uniersity Street, Peoria, IL 61604, USA Received 17 September 2001; received in revised form 6 February 2002; accepted 8 February 2002 Abstract The crystal structure of -D-glucopyranosyl-(1 4)--D-glucopyranose (-cellobiose) in a complex with water and NaI was determined with Mo K radiation at 150 K to R =0.027. The space group is P 2 1 and unit cell dimensions are a =9.0188, b =12.2536, c =10.9016 A , =97.162°. There are no direct hydrogen bonds among cellobiose molecules, and the usual intramolecular hydrogen bond between O-3H and O-5is replaced by a bridge involving Na + , O-3, O-5, and O-6. Both Na + have sixfold coordination. One I - accepts six donor hydroxyl groups and three CH···I - hydrogen bonds. The other accepts three hydroxyls, one Na + , and five CH···I - hydrogen bonds. Linkage torsion angles O-5 and C-5 are -73.6 and -105.3°, respectively ( H =47.1° and H =14.6°), probably induced by the Na + bridge. This conformation is in a separate cluster in , space from most similar linkages. Both C-6OH and C-6OH are gg, while the C-6OH groups from molecules not in the cluster have gt conformations. Hybrid molecular mechanics/quantum mechanics calculations show 1.2 kcal/mol strain for any of the small-molecule structures. Extrapolation of the NaI cellobiose geometry to a cellulose molecule gives a left-handed helix with 2.9 residues per turn. The energy map and small-molecule crystal structures imply that cellulose helices having 2.5 and 3.0 residues per turn are left-handed. © 2002 Elsevier Science Ltd. All rights reserved. Keywords: -Cellobiose; Cellulose; Mercerization; Modeling; QM/MM; Salt complex; Crystal structure 1. Introduction Substantial progress has been made in determining the structure of exceptionally crystalline samples of cellulose. 1 However, many questions about cellulose structure remain when it is in industrial and biological environments where it has lesser or altered crystallinity. Therefore, it is important to understand its intrinsic shape, its degree of flexibility, and the environmental effects on these properties. One way to increase this understanding is to continue to study di- and oligosac- charides as model compounds. Cellobiose, the smallest molecule that contains the linkage and repeated glucose rings of cellulose, has been studied by X-ray crystallography 2–4 in the usual - anomeric form and by NMR spectroscopy. 5 About 30 years ago, the preparation of microcrystalline -cel- lobiose was reported, along with a crystalline NaI complex. 6 However, structures were not determined. This paper reports the structure of a salt complex from that work. In addition to its implications for the shape properties of cellulose, interactions with Na + ions in this complex provide insight on mercerization, a poorly understood commercial treatment of cotton cellulose with NaOH. Because each experiment determines one, or at most a few, molecular shapes, data from other molecules that have small chemical differences from cellobiose are also useful in understanding cellulose. The variations in constitution inevitably cause differences in the crystal * Corresponding authors. Tel.: +1-504-2864410 (A.D.F.); tel.: +1-504-2806856 (E.D.S.). E -mail addresses: estevens@uno.edu (E.D. Stevens), afrench@srrc.ars.usda.gov (A.D. French). 0008-6215/02/$ - see front matter © 2002 Elsevier Science Ltd. All rights reserved. PII:S0008-6215(02)00041-1