www.ijbcp.com International Journal of Basic & Clinical Pharmacology | May 2019 | Vol 8 | Issue 5 Page 995
IJBCP International Journal of Basic & Clinical Pharmacology
Print ISSN: 2319-2003 | Online ISSN: 2279-0780
Original Research Article
Therapeutic drug monitoring of phenytoin using high performance
liquid chromatography in a tertiary care hospital of Kashmir, India
Mohd Adil*, Sameena Farhat, Mohd Younis Rather
INTRODUCTION
Therapeutic drug monitoring (TDM) is the clinical process
of measuring the level of particular drugs at defined
intervals to maintain a constant concentration in patients
body fluids (plasma, serum or saliva), thus helping in the
optimisation of individual drug therapy. Primarily TDM
has a role in drugs with narrow therapeutic indices and
marked pharmacokinetic variability. TDM is based on the
assumption that there is a significant relationship between
dose and body fluid concentration, and between
concentration and therapeutic effects.
1
Phenytoin is one of the most widely prescribed first line
antiepileptic agents in the Indian population.
2
Phenytoin
(PHT) is used in the treatment of primary or secondary
generalized tonic-clonic seizures, partial or complex
partial seizures and status epilepticus.
3
It is the most
commonly prescribed AED in this set-up due to its cost
effectiveness and easy availability.
4,5
ABSTRACT
Background: Phenytoin is the most commonly used anti-epileptic drug (AED)
in this set up due to cost effectiveness and easy availability. Significant
fluctuations in serum phenytoin levels leading to toxicities or treatment failures
make it an ideal candidate for therapeutic drug monitoring (TDM).
Methods: Patients of age ≥18 years who were put on phenytoin were enrolled in
this study. Estimation of serum phenytoin levels was done using HPLC. Data was
analysed using SPSS version 20.0. Chi square test, Kruskal Wallis test were used
to analyse the data.
Results: A total of 105 patients enrolled in the study, twenty patients (19%) had
normal or therapeutic serum phenytoin levels. Thirty-nine patients (37.2%) had
sub therapeutic serum phenytoin levels, while forty-six patients (43.8%) had toxic
serum phenytoin levels.
Conclusions: The TDM of phenytoin should adopt a multi-disciplinary approach
with active involvement of neuro-physicians, pharmacologists, pharmacists and
other technical staff for improving the overall management of epilepsy. TDM
data will provide the clinicians with greater insight into the factors determining
the patient’s response to drug therapy.
Keywords: Epilepsy, HPLC, Phenytoin, TDM
DOI: http://dx.doi.org/10.18203/2319-2003.ijbcp20191590
Department of Pharmacology,
Government Medical College,
Srinagar, Jammu and Kashmir
190010, India
Received: 22 February 2019
Accepted: 20 March 2019
*Correspondence to:
Dr. Mohd Adil,
Email: shahadil05@gmail.com
Copyright: © the author(s),
publisher and licensee Medip
Academy. This is an open-
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