European Journal of Pharmacology, 147 (1988) 153-154 153
Elsevier
EJP 0109R
Rapid communication
Altered haloperidol-sensitive o receptors in the genetically dystonic (dt) rat
Wayne D. Bowen *'1 j. Michael Walker 2 Alyson G. Yashar a, Rae R. Matsumoto 2
Francis O. Walker 3 and Joan F. Lorden 4
1 Sectton of Bwchemtstry, Dwlston of Btology and Medtcme, and e Walter S Hunter Laboratory of Psychology, Brown Unwersity,
Promdence, Rhode Island 02912, s Department of Neurology, Bowman Gray School of Medtcme, Wake Forest Unwerstty,
Wmston-Salem, North Carohna 27103, and 4 Department of Psychology, Unwerstty of Alabama at Bwmmgham,
Bwmmgham, Alabama 35294, USA
Recewed 21 January 1988, accepted 22 January 1988
Haloperldol-sensltlVe o receptors (Oh) are
umque non-dopamlnerglc, non-opiate receptors
found throughout many brain areas involved in
motor function. Some of the most densely popu-
lated sites include the cerebellum, red nucleus,
locus coeruleus, substantla mgra pars compacta
and select motor nuclei of spinal and cramal nerves
(Gundlach et al., 1986).
An important role of o h receptors in movement
was suggested by the potent dystomc effects of a h
hgands occurnng after nucromjectlon in the red
nucleus and the orchng behawor induced by ln-
tranigral admamstratlon of the selective o h hgand
1,3-dl-o-tolylguanldme (DTG) (Weber et al, 1986,
Walker et al., in press) Since o h receptors brad
many neuroleptlc drugs, these findings suggest
that some of the motor effects of antlpsychotlc
drugs might be mediated by o h receptors rather
than dopamlne receptors as is commonly thought
These effects further suggest that o h receptors
might be involved m dystoma, a movement dis-
order winch frequently results from neuroleptlc
drug therapy (cf Fahn, 1982) Idiopathic forms of
dystoma also occur In humans either sponta-
neously or as an lnhented disorder (Fahn, 1982).
Lorden et al. (1988) reported that Sprague-Dawley
rats with the autosomal recessive mutation (dt)
* To whom all correspondence should be addressed
exinblt severe dystonla. A mechanism lnvolwng a h
receptors was suggested by findings that these
ammals show normal doparmne, fl-adrenerglc and
muscarlnlC chohnerglc bindmg parameters, yet
they fall to become cataleptic after administration
of haloperldol (Walker et al, in press). We report
that these ammals exhibit markedly abnormal o h
binding in whole brain suggesting that defectwe
a h receptors may underhe tins and perhaps other
forms of dystoma
The brains of 4 dystomc (dt) rats and 4 normal
littermates (2 males and 2 females) were homoge-
mzed in ice-cold 10 mM Tns-HC1 pH 7 4 contain-
Ing 320 mM sucrose using a Potter-Elvehjem ho-
mogemzer with a motor-driven pestle. A crude
synaptosomal (P2) fraction was then prepared by
differential centrlfugatlon, with final resuspenslon
in 10 mM Trls-HC1 pH 7 4 at a protein concentra-
tion of 18 mg/ml Membranes (325 #g protelfi)
were incubated with 3 nM [3H]DTG and 13 con-
centraUons of unlabeled DTG ranging from 1-200
nM. Incubations were carned out in 0.5 ml of 50
mM Tns-HC1 pH 8.0 for 60 mln at 25 °C Non-
specific binding was deterrmned in the presence of
1 /zM halopendol Assays were terminated by
addition of 5 ml ice-cold 10 mM Tns-HC1 pH 7.4
and rapid filtration through glass fiber filters usmg
a Brandel Cell Harvester Filters were then washed
twice with 5 ml of buffer Filters were soaked at
least 30 mln in 0.5% polyethylenelmlne prior to
use
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