Research Article
Interaction of Ziziphus mucronata subsp. mucronata Methanol
Extract and First-Line Antibiotics is Synergistic In Vitro through
Production of Reactive Oxygen Species
Aderonke Ariyike Olajuyigbe,
1
Olufunmiso Olusola Olajuyigbe ,
2,3
and Roger Murugas Coopoosamy
3
1
Department of Biochemistry, Olabisi Onabanjo University, Ago-Iwoye, Ogun State, Nigeria
2
Department of Microbiology, School of Science and Technology, Babcock University, PMB 4005, Ilisan-Remo,
Ogun State, Nigeria
3
Department of Nature Conservation, Faculty of Natural Science, Mangosuthu University of Technology, Durban 4026,
South Africa
Correspondence should be addressed to Olufunmiso Olusola Olajuyigbe; funmijuyigbe12@yahoo.com
Received 27 December 2019; Revised 19 February 2020; Accepted 9 March 2020; Published 8 April 2020
Academic Editor: Shyam Sundar
Copyright © 2020 Aderonke Ariyike Olajuyigbe et al. is is an open access article distributed under the Creative Commons
Attribution License, which permits unrestricted use, distribution, and reproduction in any medium, provided the original work is
properly cited.
With the increased incidence of antibacterial resistance in microorganisms, combining natural products from plants with
antibiotics may be considered interesting alternatives for synergy to attain multitarget effects. In this study, the antioxidant activity
of the methanol extract of Ziziphus mucronata and its interactions with antibiotics against bacteria of clinical importance were
investigated. While its phytochemicals and antioxidant activities were determined by free radical scavenging assays, the anti-
bacterial activities of the extract and its interactions with the antibiotics were determined by macrobroth dilution and the
checkerboard methods. From the results, total phenolic content was 29.67 ± 1.90 mg GAE/100 g, total flavonoid content was
8.72 ± 0.08 mg QE/100 g, and total proanthocyanidin content was 1.94 ± 0.00 mg CE/100 g of dry plant material. e inhibition
concentration 50% (IC
50
) of DPPH, BHT, and ascorbic acid was equal to 0.04 ± 0.02 mg/ml, respectively. ose of the ABTS, BHT,
and ascorbic acid were equal to 0.02 ± 0.02, 0.04 ± 0.03, and 0.04 ± 0.02 mg/ml, respectively. e checkerboard assay showed that
combining the extract with different antibiotics resulted in synergistic (38.75%), indifferent (30%), additive (28.75%), and
antagonistic (2.5%) interactions. e interactions between the extract and antibiotics resulting in enhanced antibacterial activities
could have resulted from the antioxidant activities of the extract mopping up the ROS generated by the antibiotics or the ability of
both extract and antibiotics simultaneously producing reactive oxygen species with deleterious effects resulting in synergistic
antibacterial effects.
1. Introduction
Forming the basis for practicing sophisticated ethno-
medicine and providing excellent leads for new drug
developments [1], the therapeutic significance of medic-
inal plants has become a popularized knowledge well
disseminated by virtue of their use in the treatment of
microbial infections [2]. While the medicinal properties of
many plants have been reported [3] and pharmacological
activities are due to the bioactive compounds present in
them [4], the therapeutic failures of the drugs available
today, the scarcity of novel antibiotics [5], emergence of
resistant pathogens, adverse effects and limited spectrum
of action of the currently available drugs [6], and high
level of toxicity and carcinogenicity associated with
synthetic antioxidants such as butylated hydroxytoluene
(BHT) and tert-butyl hydroquinone (TBHQ) [7] have
propelled the need to focus attention on discovering new
and better antimicrobial and antioxidant agents of plant
origin.
Hindawi
Journal of Tropical Medicine
Volume 2020, Article ID 4087394, 9 pages
https://doi.org/10.1155/2020/4087394