Research Article
A DFT Study of Structural and Bonding Properties of Complexes
Obtained from First-Row Transition Metal Chelation by
3-Alkyl-4-phenylacetylamino-4,5-dihydro-1H-1,2,4-triazol-5-one
and Its Derivatives
Hubert Jean Nono,
1
Désiré Bikélé Mama,
2
Julius Numbonui Ghogomu,
1
and Elie Younang
3
1
Department of Chemistry, Faculty of Science, University of Dschang, P.O. Box 67, Dschang, Cameroon
2
Department of Chemistry, Faculty of Science, University of Douala, P.O. Box 24157, Douala, Cameroon
3
Department of Inorganic Chemistry, Faculty of Science, University of Yaound´ e I, P.O. Box 812, Yaound´ e, Cameroon
Correspondence should be addressed to D´ esir´ e Bik´ el´ e Mama; bikelemama@yahoo.fr
and Julius Numbonui Ghogomu; ghogsjuju@hotmail.com
Received 12 December 2016; Accepted 3 May 2017; Published 3 July 2017
Academic Editor: Konstantinos Tsipis
Copyright © 2017 Hubert Jean Nono et al. Tis is an open access article distributed under the Creative Commons Attribution
License, which permits unrestricted use, distribution, and reproduction in any medium, provided the original work is properly
cited.
Density functional calculations were used to explore the complexation of 3-alkyl-4-phenylacetylamino-4,5-dihydro-1h-1,2,4-
triazol-5-one (ADPHT) derivatives by frst-row transition metal cations. Neutral ADPHT ligand and mono deprotonated ligands
have been used. Geometry optimizations have been performed in gas-phase and solution-phase (water, benzene, and N,N-
dimethylformamide (DMF)) with B3LYP/Mixed I (LanL2DZ for metal atom and 6-31+G(d,p) for C, N, O, and H atoms) and
with B3LYP/Mixed II (6-31G(d) for metal atom and 6-31+G(d,p) for C, N, O, and H atoms) especially in the gas-phase. Single
points have also been carried out at CCSD(T) level. Te B3LYP/Mixed I method was used to calculate thermodynamic energies
(energies, enthalpies, and Gibb energies) of the formation of the complexes analyzed. Te B3LYP/Mixed I complexation energies
in the gas phase are therefore compared to those obtained using B3LYP/Mixed II and CCSD(T) calculations. Our results pointed
out that the deprotonation of the ligand increases the binding afnity independently of the metal cation used. Te topological
parameters yielded from Quantum Teory of Atom in Molecules (QTAIM) indicate that metal-ligand bonds are partly covalent.
Te signifcant reduction of the proton afnity (PA) observed when passing from ligands to complexes in gas-phase confrms the
notable enhancement of antioxidant activities of neutral ligands.
1. Introduction
In recent years, the repercussion of free radicals and reac-
tive oxygen species (ROS) in neurodegenerative disorder
is more sensitive [1–4]. Te contribution of these ROS
to the pathophysiology of myocardial reperfusion damage.
Tese ROS can be oxygen-centered radicals [5] or oxygen-
centered nonradicals [6]. Te removal of electrons from
cellular membranes by these ROS and the reaction between
these latter ones and proteins [7] provoke the alteration
of the structures of these membranes and proteins. Such
alterations justify the frailty of these cellular membranes
that expose them to be attacked by invaders (viruses and
bacteria).
Nevertheless, each cell is naturally equipped by defense
systems against any destructive efect of ROS. Tis statute of
protective mechanism against ROS in humans is attributed
to antioxidant molecules [8, 9]. In general, antioxidant
molecules (tocopherol (vitamin E), ascorbic acid (vitamin
C), carotenoids, favonoids, and polyphenols) prevent the
proliferation of free radical reactions in all cell membranes.
Tis explains the emergence of studies on the investigation
of antioxidant activities of biologically active compounds.
Tis has led to increased pressure on the need for the newer
Hindawi
Bioinorganic Chemistry and Applications
Volume 2017, Article ID 5237865, 15 pages
https://doi.org/10.1155/2017/5237865