*Corresponding author:NageswaraRao R. Neelapu
Department of Bioinformatics, School of Life Sciences, GITAM Institute of Science, GITAM University, Rushikonda campus, Visakhapatnam –
530045 (AP), India.
ISSN:0976-3031
ResearchArticle
SCREENING AND IDENTIFICATION OF DRUG TARGETS AND VACCINE CANDIDATES FOR
HELICOBACTER PYLORI STRAIN Hp26695
Amita Martin Corolina Pasupuleti, Deepthi Nammi and Nageswara Rao Reddy Neelapu*
Department of Bioinformatics, School of Life Sciences, GITAM Institute of Science, GITAM University,
Rushikonda campus, Visakhapatnam – 530045 (AP), India.
DOI: http://dx.doi.org/10.24327/ijrsr.2017.0804.0140
ARTICLE INFO ABSTRACT
Helicobacter pylori, a class 1 carcinogen colonizes stomach causing gastric carcinoma. Rising
antibiotic resistance and reinfections are drawbacks of antibiotic therapies. Alternating drugs and
vaccination may be the promising approach to prevent and treat reoccurring infections. Therefore,
there is a need for discovery of drug targets, drugs and vaccine candidates for the treatment of H.
pylori. An objective of this current study is to identify potential drug targets and suitable vaccine
candidates for H. pylori strain Hp26695 by insilico genome and proteome analysis.
Drug targets were identified initially by comparing the genomes between H. pylori and Homosapien
sapiens using RAST. RAST identified a total of 569 unique genes. These unique genes later were
subjected to non-homology and gene property analysis to identify the potential drug targets.
BLASTpfollowed by gene property analysis of 569 unique genes identified seven potential drug
targets.
Vaccine candidates were identified initially by screening protein sequences for pathogenic factors.
These pathogenic factors were screened to identify non-homologous molecules and secondary
structure patterns (helices). The proteins ≤ 3 helices are subjected to screening of antigenic nature
followed by allergenicity. The proteins qualifying the above criteria were screened for antigens, B-
cells and T-cell epitopes. Proteins showing positive predictions for antigenic, B-cell, T-cell activities
are thus shortlisted as vaccine candidates for vaccine designing. Analysis identified 16 immunogenic
proteins contributing to immune-response. These methods have enabled rapid identification of
potential drug targets and vaccine candidates for strain Hp26695 with possible therapeutic
implications for gastric cancer. cancer.
INTRODUCTION
Gastric cancer is caused by infection of class 1 carcinogen
Helicobacter pylori (Zhang, 1994). Treatment for H. pylori
infection includes drugs to relieve from pain and acidity, but
not for gastritis, peptic ulcers, and gastric cancer. Carcinogenic
activity of H. pylori suggests the need for discovery of new
drug targets and drugs for prevention of H. pylori. Laboratory
techniques and bioinformatics approaches are used to identify
drug targets which can influence growth, colonization and
virulence of H. pylori(Neelapuet al., 2014). Availability of the
complete H. pylori genome sequence of pathogens provides us
the platform and opportunity to mine the genome and harness
the potential drug targets. Comparative genomic analysis
between host and pathogen would provide us with a
tremendous amount of information that can be useful in drug
target identification (Neelapuet al., 2013).Comparative
genomics analysis of host with pathogens revealed potential
drug targets in Staphylococcus aureus (Uddinet al., 2014), H.
pylori (Neelapu and Pavani, 2013; Neelapuet al.,
2015;Nammiet al., 2016)Listeria monocytogenes(Hossainet al.,
2013), Leishmaniainfantum(Sutharet al., 2009), L. major
(Florezet al., 2010), Mycobacterium leprae(Wiwanitkit, 2014),
Pseudomonas aeruginosa(Sakharkaret al., 2004),
Schistosomamansomi(Caffreyet al., 2009).Metabolic pathway
analysis (Sarkaret al., 2012), reverse docking (Caiet al., 2006)
and screening for essential genes (Duttaet al., 2006) are used to
identify drug targets in H. pylori. However, there are no
specific reports to date, on comparing genomes of H. pylori
strain Hp26695 with host Homosapiens to identify drug targets
in H. pylori. Therefore, comparing genome of host and
pathogen may provide novel drug targets for H. pylori
strainHp26695.
Available Online at http://www.recentscientific.com
International Journal of
Recent Scientific
Research
International Journal of Recent Scientific Research
Vol. 8, Issue, 4, pp. 16384-16395, April, 2017
Copyright © Amita Martin Corolinaet al, 2017, this is an open-access article distributed under the terms of the Creative
Commons Attribution License, which permits unrestricted use, distribution and reproduction in any medium, provided the
original work is properly cited.
Article History:
Received 15
th
January, 2017
Received in revised form 25
th
February, 2017
Accepted 28
th
March, 2017
Published online 28
th
April, 2017
DOI: 10.24327/IJRSR
CODEN: IJRSFP (USA)