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BRE 22185
Different epileptogenic activities of murine and
ovine corticotropin-releasing factor
F. Marrosu l, G. Mereu 2, W. Fratta 2, P. Carcangiu 2, F. Camarri 2 and G.L. Gessa 2
1Institute of Neurology and 2Institute of Pharmacology, University of Cagliari, Cagliari (Italy)
(Accepted 23 December 1986)
Key words: Corticotropin-releasing factor (CRF); Epilepsy; Naloxone; Verapamil
The behavioral and EEG effects of rat and ovine corticotropin releasing factor (r- and o-CRF) were compared. Both peptides were
injected intracerebroventricularly into rats through chronically implanted cannulae. At the doses of 0.1 and 1 ~g both peptides acti-
vated the EEG and stimulated motor activity. At the dose of 10 ~g they produced spiking activity. However, while o-CRF-induced
spiking activity was present both in the hippocampus and in the cortical leads and was associated with generalized myoclonic move-
ments, that induced by r-CRF was confined in the hippocampus and was not accompanied by myoclonic movements. Spiking activity
induced by r-CRF was suppressed by verapamil, but was not influenced by naloxone.
Experimental evidence suggests that corticotro- the rat peptide (r-CRF) in releasing ACTH from the
pin-releasing factor (CRF) 15 controls not only the rat pituitary in vitro 12.
release of adrenocorticotropin hormone (ACTH) Since, however, the two peptides differ in 7 ami-
and fl-endorphin from pituitary 6'18 but also plays a noacid positions 12, it was of interest to compare their
transmitter role in the central nervous system behavioral and EEG effects. Moreover, in order to
(CNS) 1°. obtain some information about the possible role of
In fact, in addition to CRF-immunoreactive neu- opioids and Ca 2+ in CRF action, the effect of nalox-
rons projecting to the median eminence 14, a number one and verapamil on CRF-induced seizure activity
of such neurons are widely but selectively distributed was studied.
in different brain areas 4"18. CRF has predominantly Male Sprague-Dawley rats weighing 250-300 g,
excitatory action on various neuronal populations, individually housed in a temperature controlled
both in vivo and in brain slices )'5"19. Moreover the in- room, with 12 h light-dark cycle, were used. The ani-
tracerebroventricular (i.c.v.) injection of CRF to mals were anesthetized with chloral hydrate (400
rats has been shown to produce EEG activation and mg/kg, i.p.). A 23-gauge stainless steel guide cannula
epileptic activity 5. The latter is either restricted with- was lowered into a lateral ventricle (P 1.0, V 1.6, V
in the amygdala and hippocampus or spreads from 4.6, Pellegrino-Cushman Atlas) and a dummy stylet
these regions to cortical areas H3. was positioned into the cannula. Bipolar stainless-
Associated with the electrographic seizure activi- steel electrodes were positioned in dorsal hippocam-
ty, behavioral seizure activity has been observed, pus (P 3.5, V 2.2, V 3.3, bregma being the landmark)
ranging from myoclonic movements to apparent loss and stainless-steel screw electrodes in the calvarium
of consciousness 5. over the frontoparietal and parieto-occipital cortices.
On the basis of these data, it has been suggested Electrodes were connected to a multi-pin connector
that CRF might play an important role in epilepsy 5'2°. which was anchored to the skull with dental acrylic
In the above studies the synthetic ovine peptide cement and stainless steel screws. The connection
(o-CRF) has been used, which is equally potent to between the connector and the EEG machine was
Correspondence." G.L. Gessa, Institute of Pharmacology, University of Cagliari, Via Porcell, 4, 09100 Cagliari, Italy.
0006-8993/87/$03.50 © 1987 Elsevier Science Publishers B .V. (Biomedical Division)