Pemra Raju et al,. Int J Indig Herbs Drugs 2021;6(2):49-57
49
International Journal of
Indigenous Herbs and Drugs
Open Access ISSN: 2456-7345
Development and Validation of New Analytical Method for The Simultaneous
Estimation of Darunavir And Ritonavir in Pharmaceutical Dosage Form
Pemra Raju*
1
, K. Thejomoorthy
2
, P.Sreenivasa Prasanna
3
1 Department of Pharmaceutical analysis, M.L.College of Pharmacy, S. Konda-523101.
2 Head, Department of Pharmaceutical analysis, M.L.College of Pharmacy, S. Konda-523101.
3 Principal, M.L.College of Pharmacy, S.Konda-523101.
Article Info : Abstract
Article History
Received on: 03-03-2021
Revised on : 1-04-2021
Accepted on : 25-04-2021
Keywords:
Darunavir, Ritonavir,
RP-HPLC.
A simple, Accurate, precise method was developed for the simultaneous estimation of the
Darunavir and Ritonavir in Tablet dosage form. The chromatogram was run through Agilent
C18 150 x 4.6 mm, 5m. Mobile phase containing Buffer 0.1% Formic acid: Acetonitrile, taken
in the ratio 70:30 was pumped through the column at a flow rate of 0.95 ml/min. The
temperature was maintained at 30°C. The optimized wavelength selected was 293 nm. The
retention times of Darunavir and Ritonavir were found to be 2.369min and 2.911. %RSD of
the Darunavir and Ritonavir were and found to be 0.7 and 0.5 respectively. %Recovery was
obtained as 99.67% and 99.78% for Darunavir and Ritonavir respectively. LOD, LOQ values
obtained from regression equations of Darunavir and Ritonavir were 1.49, 5.191and 0.37,
1.11 respectively. Regression equation of Darunavir is y = 5421x + 640.7, and y = 3870.x +
5191 of Ritonavir. Retention times were decreased and run time was decreased, so the
method developed was simple and economical that can be adopted in regular Quality control
tests in Industries.
Introduction
Pharmaceutical products formulated with more than one
drug, typically referred to as combination products. These
combination products can present daunting challenges to
the analytical chemist responsible for the development
and validation of analytical methods. The development
and validation of analytical methods Spectrophotometric,
High performance liquid chromatography (HPLC) and
High-performance thin layer chromatography (HPTLC) for
drug products containing more than one active ingredient.
The official test methods that result from these processes
are used by quality control laboratories to ensure the
identity, purity, potency, and performance of drug
products. The number of drugs introduced into the market
is increasing every year. These drugs may be either new
entities or partial structural modification of the existing
ones. Very often there is a time lag from the date of
introduction of a drug into the market to the date of its
inclusion in pharmacopoeias. This happens because of the
possible uncertainties in the continuous and wider usage
of these drugs, reports of new toxicities (resulting in their
withdrawal from the market), development of patient
resistance and introduction of better drugs by
competitors. Under these conditions, standards and
analytical procedures for these drugs may not be available
in the pharmacopoeias. It becomes necessary, therefore to
develop newer analytical methods for such drugs
3
Darunavir [1] (DRV) is chemically (3R,3aS,6aR)-
hexahydrofuro[2,3-b]furan-3-yl N-[(2S,3R)- 3-hydroxy-4-
[N-(2-methylpropyl)4- aminobenzenesulfonamido]-1-
phenylbutan2yl] carbamate Figure 1. It is a protease
inhibitor used to treat HIV. It acts on the HIV aspartyl
protease which the virus needs to cleave the HIV
polyprotein into its functional fragments
This article is licensed under a Creative Commons Attribution-Non Commercial 4.0 International License.
Copyright © 2021 Author(s) retain the copyright of this article.
*Corresponding Author
Pemra Raju
Email: mlcollegeofpharmacy@gmail.com
Doi: https://doi.org/10.46956/ijihd.vi.157
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