Reviews and Accounts ARKIVOC 2012 (i) 491-545
Page 491
©
ARKAT-USA, Inc
Synthesis and applications of bipyrazole systems
Bakr F. Abdel-Wahab
a
and Kamal M. Dawood
b*
a
Applied Organic Chemistry Department, National Research Centre, Dokki, Giza, Egypt
b
Chemistry Department, Faculty of Science, Cairo University, Giza 12613, Egypt
E-mail: dr
-
dawood@yahoo.com
Abstract
This review focuses on the synthetic methodologies towards ten main classes of bipyrazole
systems (according to the type of connection between them): 1,1'-, 1,3'-, 1,4'-, 1,5'-, 3,3'-, 3,4'-,
3,5'-, 4,4'-, 4,5'- and 5,5'-junctions. The research and industrial applications of these
bipyrazoles are reported as well.
Keywords: Pyrazoles, bipyrazoles, synthesis, cycloaddition, heterocycles
Table of Contents
1. Introduction
2. Synthesis and Reactions of Bipyrazoles
2.1. 1,1'-Bipyrazoles
2.2. 1,3'-Bipyrazoles
2.3. 1,4'-Bipyrazoles
2.4. 1,5'-Bipyrazoles
2.5. 3,3'-Bipyrazoles
2.6. 3,4'-Bipyrazoles
2.7. 3,5'-Bipyrazoles
2.8. 4,4'-Bipyrazoles
2.9. 4,5'-Bipyrazoles
2.10. 5,5'-Bipyrazoles
3. Applications of Bipyrazoles
4. References
1. Introduction
Three main types of connections between two pyrazole moieties can be considered; N,N-,
C,N-, and C,C-linked bipyrazoles. According to numbering there are pertinent ten systems of
bipyrazole which differ in the position of the bond between the two pyrazole rings as shown
in Figure 1.